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1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]ethan-1-one
1-cyclopentanecarbonyl-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}piperidine-4-carboxamide
4-methoxy-N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylbenzamide
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-2-(pyridin-4-ylsulfanyl)ethan-1-one
2-{2-benzyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}propanamide
5-chloro-N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-2-carboxamide
N-methyl-2-(methylsulfanyl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,3-thiazole-4-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-[2-(5-methylfuran-2-yl)ethyl]benzamide
(3R)-1-{[2-(4-chlorophenyl)-5,8-dimethoxyquinolin-3-yl]methyl}pyrrolidin-3-ol
5-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidine-1-carbonyl]-1-methyl-1H-pyrrole-3-carbonitrile
2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]ethan-1-one
3-[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
methyl 4-{[(2-{1-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-5-oxopyrrolidin-2-yl}ethyl)amino]methyl}benzoate
3-[4-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperazin-1-yl]-1λ6-thiolane-1,1-dione
{4-[(3-methoxyphenyl)methyl]-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-4-yl}methanol
2-ethyl-N-[1-(2-methoxyphenyl)propan-2-yl]-N,4-dimethyl-1,3-oxazole-5-carboxamide
(1R,5S,6R)-N-(1,2-oxazol-3-ylmethyl)-3-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxamide
2-[ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})amino]-2-(4-methoxy-3,5-dimethylphenyl)acetic acid
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-5-propyl-1,2-oxazole-4-carboxamide
N-propyl-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
2-{4-[(2,8-dimethylquinolin-4-yl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
5-[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidine-1-carbonyl]-2-(2-methyl-1,3-thiazol-4-yl)pyrimidin-4-ol
3-(4-methoxyphenyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-3-phenylpropanamide
{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(furan-2-ylmethyl)(prop-2-yn-1-yl)amine
7-methoxy-3-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-2,3,4,5-tetrahydro-1H-3-benzazepine
1-(4-{[3-(4-tert-butylbenzoyl)piperidin-1-yl]methyl}phenyl)imidazolidin-2-one
5-{2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}-4-phenyl-1H-imidazole
4-methyl-N-(oxolan-2-ylmethyl)-2-(propan-2-yl)-N-(thiophen-3-ylmethyl)-1,3-thiazole-5-carboxamide
8-(2-methylpyrimidin-4-yl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
3-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-1-(2-methylphenyl)urea
1-[2-(2,2-diphenylethyl)morpholine-4-carbonyl]cyclopropan-1-amine
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
3-[2-(dimethylamino)ethyl]-1-ethyl-8-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[3-(3-methylphenoxymethyl)piperidine-1-carbonyl]-1H-indazole
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-(oxan-3-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-[(5-ethylpyridin-2-yl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
N-methyl-2-[(prop-2-en-1-yl)amino]-N-(1H-pyrazol-5-ylmethyl)benzamide
9-[2-(ethylsulfanyl)propanoyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-ethyl-5-[1-(2-methanesulfonylethyl)-4-phenyl-1H-imidazol-5-yl]-1H-1,2,4-triazole
3-{5-[1-(pyridin-2-ylmethyl)-1H-1,2,3-triazol-4-yl]thiophen-3-yl}prop-2-yn-1-ol
1-methyl-4-{1H-pyrazolo[3,4-b]pyridin-4-yl}-1H-pyrrolo[2,3-b]pyridine
N3-{2-[(2-chlorophenyl)formamido]ethyl}piperidine-1,3-dicarboxamide
N-({1-[ethyl(methyl)amino]cyclopentyl}methyl)-4-(pyrrolidin-1-ylmethyl)benzamide
N-benzyl-5-(6-fluoro-1H-1,3-benzodiazol-2-yl)pyrimidin-2-amine
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
8-(3-hydroxy-4-methylbenzoyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
8-[(2-aminopyridin-3-yl)methyl]-2-cyclopropanecarbonyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-methoxy-4-{[methyl({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amino]methyl}phenol
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(4H-1,2,4-triazol-4-yl)ethan-1-one