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N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-3-(morpholin-4-yl)propanamide
1-(3-methylpyridin-2-yl)-4-[(2,3,4-trimethoxyphenyl)methyl]piperazine
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]propane-1-sulfonamide
(1S,5R)-3-[1-(7-fluoroquinazolin-2-yl)piperidin-4-yl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[1-(3-phenylpropyl)-5-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperazin-2-one
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
N,5-dimethyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(2S,4S)-4-amino-1-(4-cyanobenzenesulfonyl)-N,N-diethylpyrrolidine-2-carboxamide
N-methyl-2-[N-methyl-1-(2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazol-4-yl)formamido]acetamide
1-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
N-[3-(3-methylphenyl)phenyl]-1-(1H-pyrazole-4-carbonyl)pyrrolidine-2-carboxamide
(1S,3R)-3-amino-N-(3-methylcinnolin-5-yl)cyclopentane-1-carboxamide
4-{3-[methyl(1-methylpyrrolidin-3-yl)amino]propanoyl}-1-(4-methylphenyl)piperazin-2-one
2-({[2-(dimethylamino)ethyl][(2-methylphenyl)methyl]amino}methyl)benzoic acid
2-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-5-(1,2,3,4-tetrahydroisoquinolin-2-yl)-2,3-dihydropyridazin-3-one
{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}(thiophen-2-yl)methanol
methyl (2S,4S,5R)-5-(3-chlorophenyl)-1-methyl-4-[(pentan-3-yl)carbamoyl]pyrrolidine-2-carboxylate
N-methyl-2-(3-methyl-1,2-oxazol-5-yl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
(3S)-4-[(2-chloro-5-fluorophenyl)methyl]-3-ethylmorpholine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N2-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-N1-(3-methylpyridin-2-yl)ethane-1,2-diamine
({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)(quinolin-2-ylmethyl)amine
6-{2-[2-(3-hydroxyphenyl)ethyl]piperidine-1-carbonyl}-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
2-(2-chloropyridine-4-carbonyl)-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
N-(2-chlorophenyl)-2-{8-methyl-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}-2-oxoacetamide
(4aS,7aR)-1-(3,4-difluorobenzoyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
({3-methoxy-2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
9-(cyclopropylmethyl)-1-methyl-4-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(methoxymethyl)-N-methyl-N-[1-(pyridin-3-yl)propyl]cyclobutane-1-carboxamide
N-(5-aminopentyl)-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
N-cyclopentyl-1-{1,3-dioxo-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
9-[6-amino-2-(methylsulfanyl)pyrimidin-4-yl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-benzyl-N-(2-hydroxyethyl)-3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
N-(2-aminoethyl)-2-{[(2E)-3-phenylprop-2-en-1-yl]sulfanyl}pyridine-3-carboxamide
N2-[2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-N1-(pyridin-3-yl)ethane-1,2-diamine
1,4-dimethyl-2-({1-[3-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}methyl)piperazine
2-methoxy-1-{4-[2-(4-phenylpiperazine-1-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
2-(dimethylamino)-2-(4-methylphenyl)-N-[1-(morpholin-4-ylmethyl)cyclopentyl]acetamide
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-benzyl-3-[1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)piperidin-4-yl]-N-methylpropanamide
2-{[5-(3-cyclopropyl-1H-pyrazol-5-yl)-4-methyl-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
methyl 4-{[4-(1-methylpiperidin-4-yl)piperidin-1-yl]methyl}thiophene-2-carboxylate
2-methyl-4-{3-[3-(pyridin-3-yl)azetidine-1-carbonyl]phenyl}butan-2-ol
2-ethoxy-1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
5-[4-(2-methylphenyl)piperazine-1-carbonyl]-1,3-benzothiazol-2-amine
(3S,4S)-1-[3-(3-methoxyphenyl)propanoyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
6-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]pyridine-2-carbonitrile
N-{[2-(4-acetylpiperazin-1-yl)-5,8-dimethoxyquinolin-3-yl]methyl}-3-chloro-N-(oxolan-2-ylmethyl)benzamide
[2-ethoxy-5-({[(2-methylphenyl)methyl](prop-2-en-1-yl)amino}methyl)phenyl]methanol
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide