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3-(cyclopropylmethyl)-1-(2,6-difluorophenyl)-3-(2-methoxyethyl)urea
N-(3-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}phenyl)propanamide
1-(cyclopropylmethyl)-4-(4-methyl-1,3-oxazole-5-carbonyl)-2-(propan-2-yl)-1,4-diazepane
[(3R,4R)-1-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N,2-dimethyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-1,3-thiazole-5-carboxamide
N-[(4,6-dimethylpyridin-3-yl)methyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
N-[3-(1,3-benzoxazol-2-yl)propyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
2-(9H-carbazol-3-yl)-1-[(3R,4S)-4-(dimethylamino)-3-(3-hydroxypropyl)piperidin-1-yl]ethan-1-one
3-(2H-1,3-benzodioxol-5-yl)-N-(2-methoxyethyl)-N-methyl-3-phenylpropanamide
1-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-3-[3-ethyl-4-(4-fluorophenyl)-1-methyl-1H-pyrazol-5-yl]urea
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-8-methoxy-N-(propan-2-yl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-4-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazole
N-(3-phenylpropyl)-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-(2,5-dioxoimidazolidin-1-yl)-N-(oxolan-2-ylmethyl)-N-(2-phenoxyethyl)acetamide
(3R,4R)-4-amino-1-({5-chloro-2-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)piperidin-3-ol
3-methoxy-5-{pyrazolo[1,5-a]pyridin-7-yl}pyridine
2-(dimethylamino)-N,4-dimethyl-N-[1-(pyridin-2-yl)propyl]pyrimidine-5-carboxamide
3-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzonitrile
N-cyclohexyl-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]-N-(prop-2-yn-1-yl)acetamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-4-(4-methoxyphenoxy)benzamide
2-[3-(2-fluorophenoxymethyl)piperidine-1-carbonyl]-N,N-dimethylaniline
1-[(3-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-2,5-dimethylphenyl)methyl]-4-methylpiperazine
1-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]ethan-1-one
N-(2,3-dihydro-1H-inden-2-yl)-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
1-methyl-N-(pyridin-4-ylmethyl)-5-{[2-(thiophen-2-yl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(4-{[(5-ethylpyrimidin-2-yl)amino]methyl}piperidin-1-yl)ethan-1-one
2-[4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazolin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
2-(4-fluorophenyl)-1-[1-(methoxymethyl)cyclobutanecarbonyl]piperidine
2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-N-(thiophen-2-ylmethyl)aniline
1-{5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}piperidin-4-ol
2-(2-methyl-1,3-thiazol-4-yl)-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]acetamide
2,4-dimethyl-7-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]quinoline
methyl 4-[(2R,3R)-3-(dimethylamino)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-4-oxobutanoate
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-2-(4-phenylpiperidin-1-yl)acetamide
2-(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-1-(propan-2-yl)-1H-imidazole
2-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-5-fluoropyrimidine
2-(2-methoxyethyl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1,3-benzoxazole-6-carboxamide
N-cyclopropyl-4-(morpholin-4-yl)-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)benzamide
N-cyclopropyl-N-[(4-hydroxyphenyl)methyl]-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
(3aS,6aS)-2-benzyl-5-[(dimethyl-1,2-oxazol-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-[(2,5-dimethoxyphenyl)methyl]-3-(2-methylpropyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
4-[(2R)-2-{[1-(2-amino-6-methylpyrimidin-4-yl)piperidin-4-yl]amino}-3-hydroxypropyl]phenol
1-{2-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-2-oxoethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
1-amino-N-{2-[4-(2-methylpropyl)morpholin-2-yl]ethyl}cyclopentane-1-carboxamide
N-methyl-N-[(2-methylpyridin-4-yl)methyl]-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
5-propyl-3-[2-(pyridin-2-yl)ethyl]-5-{1-[2-(thiophen-3-yl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
1-(4-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
4-[({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)methyl]benzene-1-sulfonamide
N-[2-(1,3-benzoxazol-2-ylsulfanyl)ethyl]-4-chloro-1-ethyl-1H-pyrazole-3-carboxamide