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3-[3-(3-hydroxypiperidin-1-yl)propyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-N-[1-(pyridin-3-yl)propan-2-yl]pyridin-2-amine
2-{4-methyl-6-[4-(thiomorpholin-4-yl)piperidin-1-yl]pyrimidin-2-yl}phenol
3-[(3R,4S)-1-(2,3-difluoro-4-methoxybenzoyl)-4-(dimethylamino)piperidin-3-yl]propan-1-ol
5-{[4-(2-methoxybenzoyl)piperazin-1-yl]methyl}quinoxaline
6-fluoro-3-[(5-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-3,4-dihydroquinazolin-4-one
6-(4-phenylazepan-1-yl)-9H-purine
3-(3-fluorophenyl)-1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
10-methoxy-5-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-[(2-methoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)pyridine-4-carboxamide
2,2-dimethyl-N-(2-{[(3-methylphenyl)methyl]carbamoyl}phenyl)-4-oxo-3,4-dihydro-2H-pyran-6-carboxamide
(3aR,7aS)-2-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
2-[4-(1H-indol-2-ylmethyl)-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(furan-3-ylmethyl)piperidin-3-yl]propanamide
N-{[(2S,4S)-4-fluoro-1-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]pyrrolidin-2-yl]methyl}methanesulfonamide
({5-[1-(3,5-difluoropyridine-2-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
8-(6-methylpyridine-2-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
3,5-dimethyl-4-oxo-N-[(2R)-pyrrolidin-2-ylmethyl]-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
1-[2-(1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-3-(3-hydroxyquinoxalin-2-yl)propan-1-one
({2-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]phenyl}methyl)dimethylamine
[(3,5-dichloropyridin-4-yl)methyl](methyl)[2-(oxan-2-yl)ethyl]amine
(3aS,6aS)-2-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-5-(2-hydroxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propan-2-ol
N-[(1-benzylpyrrolidin-3-yl)methyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[3-(5-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]ethan-1-one
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-4-carboxamide
N-[2-(cyclohexylsulfanyl)ethyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-4-(piperidin-3-yl)benzamide
3-(4-benzyl-1H-pyrazol-5-yl)-1-(1-methyl-1H-pyrazole-4-carbonyl)piperidine
3-chloro-N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-6-methylpyrazolo[1,5-a]pyrimidine-2-carboxamide
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-N-(furan-2-ylmethyl)piperidine-1-carboxamide
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(benzenesulfonyl)-2,8-diazaspiro[4.5]decane-2-carboxamide
1,4,6-trimethyl-N-[(1-methylpiperidin-3-yl)methyl]-2-oxo-N-(2-phenylethyl)-1,2-dihydropyridine-3-carboxamide
(2R,6R)-4-(2,4-dimethylpyrimidine-5-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]urea
N-{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}-N-methyloxolan-3-amine
1-({[2-(5-cyano-2-methyl-1H-indol-3-yl)ethyl]carbamoyl}methyl)piperidine-4-carboxamide
1-(8-methylquinolin-5-yl)-3-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}urea
2-{4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}acetamide
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-6-oxo-1,6-dihydropyrimidine-5-carboxamide
1-[2-(1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
N-[2-(4-chlorophenyl)ethyl]-2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}acetamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-[5-oxo-2-(thiophen-2-yl)cyclopent-1-en-1-yl]acetamide
1-[3-(8-methoxyquinolin-5-yl)-4-(morpholin-4-yl)phenyl]ethan-1-one
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(oxan-4-yl)piperidine-3-carboxamide
3-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-1-(3-methyl-1,2,4-thiadiazol-5-yl)urea
4-(3-aminopiperidine-1-carbonyl)-1,2-dihydroisoquinolin-1-one
6-(oxolan-2-yl)-3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
2-({1-[(3-methoxyphenyl)methyl]piperidin-3-yl}amino)pyridine-3-carboxylic acid