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(2S,4R)-4-amino-N-ethyl-1-[1-(3-methylbutanoyl)piperidine-4-carbonyl]pyrrolidine-2-carboxamide
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(pyridin-3-ylmethyl)pyridin-2-amine
2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
2-[5-(2-methoxypyridin-3-yl)-1H-indazol-1-yl]-N-(1-methyl-1H-1,2,3-triazol-4-yl)acetamide
6-ethyl-4-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1,2-dihydropyridin-2-one
3-(5-{2-[2-(2-methyl-1,3-oxazol-4-yl)-1H-imidazol-1-yl]ethyl}-1H-1,2,4-triazol-3-yl)pyridine
N-[1-(pyrazin-2-yl)piperidin-4-yl]-3-(1H-pyrazol-1-ylmethyl)benzamide
N-[2-(1H-imidazol-1-yl)ethyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
1-methyl-2-oxo-8-{[2-(trifluoromethyl)phenyl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(4-tert-butylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-ethyl-N-{[2-(3-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]butanamide
2-methyl-3-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-4,5,6,7-tetrahydro-2H-indazole
6-amino-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methylpyridine-2-carboxamide
methyl[2-(morpholin-4-yl)ethyl]{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
4,4,4-trifluoro-1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}butan-1-one
1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(1H-pyrazol-1-yl)butan-1-one
4-(5-chloropyrimidin-2-yl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
8-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3,5-dimethyl-2-[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidine-1-carbonyl]-1H-indole
5-ethyl-2-{1-[2-(1H-imidazol-4-yl)ethyl]-1H-1,2,3-triazol-4-yl}pyridine
(3aS,7aR)-5-methyl-2-(5-propylpyrimidin-4-yl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
N,N-dimethyl-7-(oxolane-3-carbonyl)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}-2-(1H-pyrazol-1-yl)butan-1-one
4-(1-butyl-1H-imidazol-2-yl)-1-(2,6-difluorobenzoyl)piperidine
3-[(4-methoxyphenyl)methyl]-5-(pyrrolidin-1-ylmethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
N-(1-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N,2-dimethylfuran-3-carboxamide
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]thian-4-amine
4-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)-1-(thian-4-yl)piperidine
3-{[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidin-1-yl]methyl}-7-fluoro-1,2-dihydroquinolin-2-one
N-[(3S,4R)-1-[(4-oxo-4H-chromen-3-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
1-(3-methyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-4-(2-methylquinolin-6-yl)piperidin-4-ol
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-(2-hydroxyethyl)-N-(1,3-thiazol-2-ylmethyl)butanamide
4-[(2-methylphenyl)methyl]-1-[4-(piperidin-1-ylmethyl)benzoyl]-1,4-diazepan-5-one
(2S,4R)-1-benzyl-N-methyl-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-amido}pyrrolidine-2-carboxamide
1-[4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
N-[(2R,4R,6S)-2-tert-butyl-6-(6-chloro-2-fluoro-3-methoxyphenyl)oxan-4-yl]acetamide
4-[4-(hydroxymethyl)benzoyl]-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
{9-methyl-3-[2-(1H-pyrazol-4-yl)ethyl]-3,9-diazaspiro[5.5]undecan-1-yl}methanol
6-(4-methoxyphenyl)-9-[2-(methylsulfanyl)pyridine-3-carbonyl]-6,9-diazaspiro[4.5]decan-7-one
3-(1-{[1-(4-chlorophenyl)propan-2-yl]amino}ethyl)adamantan-1-ol
1-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
1-{2-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-2,7-diazaspiro[4.5]decan-7-yl}-3-methoxypropan-1-one
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
4-benzyl-3-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-4-methyl-N-(2-methylpropyl)-1,2,3-thiadiazole-5-carboxamide
4-({4-methyl-5-[1-(2-methylpyrimidin-4-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
ethyl 2-(1-{3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]phenyl}-N-methylformamido)acetate
1-[4-(piperidine-1-carbonyl)piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-amine