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2-{3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-4-methylpyrimidine
2-(2-methyl-1,3-thiazol-4-yl)-5-{3-oxa-9-azaspiro[5.5]undecane-9-carbonyl}pyrimidin-4-ol
4,4,4-trifluoro-1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]butan-1-one
2-{3-[1-(oxan-4-ylmethyl)-1H-1,2,3-triazol-4-yl]phenoxy}acetamide
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}pyrazine-2-carboxamide
1-[1-(7-chloroquinolin-4-yl)piperidin-4-yl]piperidin-4-ol
1-(2-methylpyridin-4-yl)-4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-1,4-diazepane
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
6-chloro-2-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
4-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl}benzene-1-sulfonamide
1-[6-(2-ethylphenyl)pyridine-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
N-[(1-hydroxycyclohexyl)methyl]-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
(2S,4R)-4-(3-cyanobenzamido)-N,N-diethyl-1-propanoylpyrrolidine-2-carboxamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-[2-(1H-imidazol-4-yl)ethyl]-1H-pyrazole-3-carboxamide
1-{5-[2-(furan-2-yl)azepane-1-carbonyl]thiophen-2-yl}ethan-1-one
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
4-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
6-chloro-4-[2-(trifluoromethyl)morpholin-4-yl]quinoline
(2S)-N-(2,4-dichloro-3-methylphenyl)-2-(methoxymethyl)pyrrolidine-1-carboxamide
(2-{[(1,3-dimethyl-1H-pyrazol-5-yl)methyl][(2-methylphenyl)methyl]amino}ethyl)dimethylamine
2-{4-[(4-methoxyphenyl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-(1H-indol-4-ylmethyl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-methyl-N-(1,2-oxazol-5-ylmethyl)-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
(4aS,7aR)-1-(2-chlorobenzoyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6,7-dimethoxy-2-(3-propyl-1H-pyrazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinoline
6-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine-3-carboxylic acid
N-cyclohexyl-2-(4-ethyl-2,3-dioxopiperazin-1-yl)-N-(thiophen-3-ylmethyl)acetamide
4-(1-{[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}azetidin-3-yl)morpholine
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl][(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(pyridin-3-yl)propanamide
6-[2-(morpholin-4-ylmethyl)phenyl]quinoline
(2S,4R)-1-[(2-chloro-6-fluorophenyl)methyl]-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
methyl 3-(cyclobutylmethoxy)-5-[(3S)-3-(dimethylamino)pyrrolidine-1-carbonyl]benzoate
N-[(3S)-1-benzylpyrrolidin-3-yl]-N-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
6-methyl-1-{3-oxo-3-[4-(1,3-thiazol-2-yl)piperazin-1-yl]propyl}-1,2-dihydropyridin-2-one
1-[2-(methylsulfanyl)pyrimidin-4-yl]-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]piperidin-4-amine
4-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methylpyridine
1-(but-2-ynoyl)-N-[4-(2-fluorophenoxy)phenyl]piperidine-2-carboxamide
4-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-ethyl-1-methylpiperazine
5-{8-chloro-[1,2,4]triazolo[4,3-a]pyridin-3-yl}-1-ethyl-1H-imidazole
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-N-methyl-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
ethyl (4aR,6R,8aS)-2-(1H-imidazol-4-ylmethyl)-6-(morpholin-4-yl)-decahydroisoquinoline-8a-carboxylate
N-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-2-(pyridin-3-yl)piperidine-1-carboxamide
methyl 2-[(3,5-dimethylphenyl)sulfamoyl]-6-(2-methylpropanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)-N-[2-(pyridin-2-yl)ethyl]quinoline-4-carboxamide
1-(1'-{imidazo[1,2-a]pyrimidine-2-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)ethan-1-one
2-(4-chlorophenyl)-4-[6-(propan-2-yl)pyrimidin-4-yl]morpholine
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
(1R,3S)-3-{[(5-methylthiophen-2-yl)methyl](pyridin-4-ylmethyl)carbamoyl}cyclopentane-1-carboxylic acid