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1-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(methylsulfanyl)propan-1-one
1-[1-(4-chlorophenyl)cyclobutaneamido]cyclopentane-1-carboxylic acid
(benzylsulfamoyl)({[2-fluoro-3-(trifluoromethyl)phenyl]methyl})amine
7-[(5-cyclopentylthiophen-2-yl)methyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-{[benzyl(1,3-thiazol-2-ylmethyl)amino]methyl}-6-methylpyridin-3-ol
4-({[6-(aminomethyl)-2-methylpyrimidin-4-yl]amino}methyl)benzene-1-sulfonamide
N-methyl-5-[1-(2-{[(2-methylphenyl)methyl]sulfanyl}acetyl)pyrrolidin-2-yl]thiophene-2-carboxamide
2-methyl-5-oxo-N-[3-(3-phenylpropoxy)phenyl]-1,4-diazepane-1-carboxamide
1-methyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydropyridin-2-one
1-(1-methyl-1H-pyrazole-5-carbonyl)-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-2,2-dimethylpropanamide
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
3-(4-methyl-1,3-thiazol-5-yl)-N-[1-(pyrazin-2-yl)propan-2-yl]propanamide
2-(methylamino)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)acetamide
4-({4-[3-(cyclopropylcarbamoyl)piperidin-1-yl]piperidin-1-yl}methyl)benzoic acid
N-{4-[2-(2-hydroxyphenyl)acetamido]-2-methylphenyl}-2,2-dimethylpropanamide
(2S,4S)-4-(2,6-difluoro-4-methoxybenzamido)-N-ethyl-1-propylpyrrolidine-2-carboxamide
N-cyclopentyl-2-(4-fluorophenyl)-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}acetamide
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1H-1,2,3-triazole-5-carboxamide
3-[(3R,4S)-1-[2-(3-fluoro-4-methylphenyl)acetyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
2-[5-(2-amino-9H-purin-6-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
(4aS,7aR)-1-(3-phenylpropyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N,4-dimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-3-(2-oxoimidazolidin-1-yl)benzamide
1-methyl-3-(2-methylpropyl)-N-[2-(1H-pyrrol-1-yl)ethyl]-1H-pyrazole-5-carboxamide
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}ethane-1-sulfonamide
1-[7-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]-2-(propan-2-yloxy)ethan-1-one
5-(2,3-dimethoxy-5-methylphenyl)-4-methylpyridin-2-amine
1-{3-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenyl}ethan-1-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}thiophene-3-carboxamide
methyl 5-cyano-2-methyl-6-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}pyridine-3-carboxylate
methyl 2-(2-methoxy-3,5-dimethylphenyl)-1H-1,3-benzodiazole-6-carboxylate
2-[4-(5,6-dimethylpyrimidin-4-yl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-(trifluoromethyl)piperidine
N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}cyclopentanamine
N-ethyl-5-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]pyrimidin-2-amine
(4aR,7aS)-1-methyl-4-(2-{2-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-ethyl-5-[3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]pyrimidin-2-amine
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(furan-2-yl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
N-methyl-3-(2-methylphenyl)-3-phenyl-N-(pyrimidin-4-ylmethyl)propanamide
2,6-dihydroxy-N-[1-(3-hydroxyadamantan-1-yl)ethyl]benzamide
N-[(3-methylphenyl)methyl]-N-(propan-2-yl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-(ethylsulfanyl)-5-[4-phenyl-1-(pyridin-3-ylmethyl)-1H-imidazol-5-yl]pyrimidine
1-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}-2-(propan-2-yloxy)ethan-1-one
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(4-phenylphenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-(4-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)ethan-1-one
1-[(3,5-dimethylphenyl)methyl]-4-(5-methoxypyrimidin-2-yl)piperazin-2-one
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-amine
2-(2,3-dimethoxyphenyl)-1-[2-(pyridin-2-yl)piperidin-1-yl]ethan-1-one
N,N-diethyl-1-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)piperidine-3-carboxamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-4-(piperidin-1-ylmethyl)benzamide