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6-amino-2-{2-[({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]ethyl}pyrimidin-4-ol
6-(5-oxo-1,4-diazepan-1-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
2-(cyclopent-2-en-1-yl)-1-[3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
3-[8-(2,3-dihydro-1H-indene-5-carbonyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl]propanoic acid
N-cyclohexyl-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]urea
2-(furan-2-ylmethyl)-9-{spiro[2.3]hexane-1-carbonyl}-2,9-diazaspiro[5.5]undecan-3-one
2-(1-methyl-1H-pyrrol-3-yl)-1-{4-[(oxolan-3-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}ethan-1-one
N-methyl-N-(2-methylpropyl)-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
N-cyclopentyl-2-{2-[3-oxo-3-(pyrrolidin-1-yl)propyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}propanamide
N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
(2S,4R)-4-(dimethylamino)-1-[(1-methyl-1H-indol-2-yl)methyl]pyrrolidine-2-carboxylic acid
9-(2-acetylbenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
(1R,3S)-3-methoxy-7-{[2-(trifluoromethoxy)phenyl]methyl}-7-azaspiro[3.5]nonan-1-ol
2-methyl-5-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1H-1,3-benzodiazole
5-[3-(3-fluorophenoxymethyl)piperidine-1-carbonyl]-2-methyl-1H-1,3-benzodiazole
N2-(2-methoxyethyl)-N4-[1-(pyrazin-2-yl)propan-2-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methylphenoxy)piperidine
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)thian-4-amine
5-chloro-3-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
2-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
6-{1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
1-[(3-methoxyphenyl)methyl]-4-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-2-one
(4S)-1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-3,3,4-trimethylpiperidin-4-ol
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
2-{3-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]piperidin-1-yl}acetamide
2-{4-[(4-fluorophenyl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
N-[2-(3-chlorophenyl)ethyl]-2-{methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}acetamide
1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,4-diazepan-5-one
N-[1-(2-chlorophenyl)cyclopropyl]-2-(methylamino)pyrimidine-5-carboxamide
6-methoxy-1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]hexan-1-one
N-[(4-fluorophenyl)methyl]-3-[1-(oxolane-2-carbonyl)piperidin-4-yl]propanamide
1-{4-[2-(4-methylpentyl)morpholine-4-carbonyl]piperidin-1-yl}ethan-1-one
N-methyl-5-(3-methyl-1,2,4-oxadiazol-5-yl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]pyridin-2-amine
1-(dimethyl-1,2-oxazole-4-carbonyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
5-[(1-benzothiophen-2-ylmethyl)(methyl)amino]-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N,N-dimethyl-4-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}-4-oxobutanamide
1-(2-fluoro-4-methoxyphenyl)-3-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}urea
4-[2-hydroxy-4-(methylsulfanyl)butanoyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
4-(4-propylbenzenesulfonyl)-2-(trifluoromethyl)morpholine
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-4-(1H-pyrazol-3-yl)benzamide
N,6-dimethyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-2-oxo-4-(pyridin-3-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
3-(2-phenoxyethyl)-8-[2-(1H-1,2,4-triazol-1-ylmethyl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
ethyl 1-{[1-(carbamoylmethyl)-1H-indol-3-yl]methyl}-4-(2-phenylethyl)piperidine-4-carboxylate
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
2-methoxy-N-({5-[3-(trifluoromethoxy)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)acetamide
3-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-[1-methyl-3-(pyridin-3-yl)-1H-pyrazol-5-yl]urea
N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
(3S,5R)-5-[(4-fluorophenyl)carbamoyl]-1-(2-hydroxypyridine-3-carbonyl)piperidine-3-carboxylic acid