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N-[(1-ethylpyrrolidin-2-yl)methyl]-3-(morpholine-4-carbonyl)benzene-1-sulfonamide
2-({4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)benzonitrile
1-benzyl-N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}pyrrolidin-3-amine
5-cyclopropanecarbonyl-1'-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-fluoro-4-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}pyridine
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
2-[4-(1,3-benzoxazol-2-yl)-1-[(3-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
3-(azocan-1-yl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]propanamide
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,2,2-trimethyloxane-4-carboxamide
N-methyl-2-[4-methyl-6-(morpholine-4-carbonyl)-3,4-dihydro-2H-1,4-benzoxazin-3-yl]-N-(prop-2-yn-1-yl)acetamide
(3aR,6aR)-2-methanesulfonyl-5-[3-(pyridin-3-yl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-chlorothiophene-2-carboxamide
N2-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-N1-(3-methylpyridin-4-yl)ethane-1,2-diamine
1-(3-methylpiperidin-1-yl)-3-({[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}amino)propan-1-one
2-(2,3-dihydro-1H-inden-2-yl)-1,2,3,4-tetrahydroisoquinolin-4-ol
3-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-2-ethyl-6-methyl-1-(thiophen-2-ylmethyl)-1,4-dihydropyridin-4-one
8-[(2-chloro-4-fluorophenyl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{[2-(difluoromethoxy)phenyl]methyl}-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
4-hydroxy-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N,5,7-trimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
8-[2-(3-chloro-4-fluorophenoxy)acetyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
[4-({4-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}methyl)phenyl]methanol
7-fluoro-N,2-dimethyl-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}quinoline-4-carboxamide
methyl (2S,4R)-1-[(2-hydroxyphenyl)methyl]-4-(2-phenylbenzamido)pyrrolidine-2-carboxylate
(4-methyl-5-{1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methanol
{[3-(4-chlorophenoxy)phenyl]methyl}({3-[4-(morpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl})amine
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[1-(thiophen-2-yl)propan-2-yl]benzamide
2-[3-chloro-5-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carbonitrile
(4aS,7aR)-4-(2-methoxyethyl)-N-(3-methoxyphenyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-{9-[2-(2-methylphenyl)acetyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
3-butanamido-4-methyl-N-{3-[(5-methylpyridin-2-yl)amino]propyl}benzamide
N-benzyl-2-(dimethyl-1,2-oxazol-4-yl)pyrrolidine-1-sulfonamide
7-(3-chlorophenyl)-4-(2,2-dimethylcyclopropanecarbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{2-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-indazol-3-one
1-[(4-methoxyphenyl)methyl]-4-(2,3,4-trifluorobenzoyl)piperazin-2-one
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine
1-[6-(4-chloro-3-fluorophenyl)pyridazin-3-yl]azepane
2-(1H-imidazol-2-yl)-1-(2,2,2-trifluoroethyl)-1H-imidazole
N-[(3-methoxyphenyl)methyl]-1-methyl-N-(prop-2-en-1-yl)-3-propyl-1H-pyrazole-5-carboxamide
2-[cyclopentyl(methyl)amino]-1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
6-butyl-2-(4-{[3-(methoxymethyl)piperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
[(3S,5R)-1-[1-(methoxymethyl)cyclopropanecarbonyl]-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
N,N,2-trimethyl-7-(1,2,3,4-tetrahydroquinoline-8-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-{2-[ethyl(3-methylphenyl)amino]ethyl}-2,5-dimethyl-1,3-thiazole-4-carboxamide
8-(1,3-benzothiazol-2-ylmethyl)-3-[2-(dimethylamino)ethyl]-1-[2-(4-methoxyphenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(5-methyl-1-propyl-1H-pyrazol-4-yl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyrimidin-2-amine
9-[6-(dimethylamino)pyrimidin-4-yl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[1-(1-methyl-1H-imidazol-2-yl)butyl]-2-(2,3,6-trimethylphenoxy)acetamide
2-[({1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)amino]acetamide