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3-ethyl-3-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-[3-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]urea
(4aS,8aR)-1-(3-methoxypropyl)-6-[3-(1H-pyrrol-1-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
2-(1-ethyl-1H-imidazol-5-yl)-7-(3-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-[4-(4-methoxyphenyl)-2-methyl-5-oxopiperazin-1-yl]-N-[(2-methylphenyl)methyl]acetamide
1-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3-(1-propyl-1H-1,2,4-triazol-3-yl)urea
2-(1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidin-3-yl)-1,3-benzothiazole
2-[3-(methoxymethyl)pyrrolidin-1-yl]-5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridine
1-ethyl-5-{2-[(2-methylphenyl)sulfanyl]acetyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-[(4aR,8aR)-7-(3-fluoro-4-methoxybenzoyl)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
4-{6-methylthieno[2,3-d]pyrimidin-4-yl}-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
3-{2-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}benzamide
2-(3-hydroxypropyl)-9-[(6-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
4-methyl-N-({1-[2-(1H-pyrazol-1-yl)ethyl]-1,2,3,6-tetrahydropyridin-4-yl}methyl)benzamide
4-(4-{methyl[(methylcarbamoyl)methyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)benzamide
N-(2-methyl-1,3-benzothiazol-6-yl)-3-(pyridine-3-carbonyl)piperidine-1-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1-[2-(2-methoxyphenyl)ethyl]-2,6-dimethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
1-(2-methoxyphenyl)-4-{1-[(5-methylfuran-2-yl)methyl]piperidin-3-yl}piperazine
methyl 3-[4-(1,3-oxazol-5-yl)benzamido]azepane-1-carboxylate
2-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-N-methylacetamide
N-(3-hydroxypropyl)-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(4-chlorophenyl)methyl]-4-{[(4-fluorophenyl)methyl]amino}pyrrolidine-2-carboxamide
1-{1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
3-hydroxy-3-{[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
4-({[(3-ethoxyphenyl)methyl](2-hydroxyethyl)amino}methyl)benzonitrile
(4aS,7aR)-1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[(2,3-difluoro-4-methylphenyl)methyl]-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-phenyl-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
5-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pent-4-en-1-one
3-{3-[1-(2-methoxyethyl)-1H-pyrazol-3-yl]phenyl}-6-(propan-2-yloxy)pyridazine
3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxy-N-[2-(methylsulfanyl)ethyl]benzamide
2-[(1-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)oxy]pyrimidine
N-[2-({2,6-dimethylimidazo[1,2-a]pyridin-3-yl}formamido)ethyl]-4-fluorobenzamide
3-(2-oxo-2-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)-1,3-oxazolidin-2-one
3-ethyl-1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-ol
3-(2-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
{[2-(morpholin-4-yl)pyridin-3-yl]methyl}(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
1-(4-acetylpiperazin-1-yl)-3-(3-methylpiperidin-1-yl)propan-1-one
4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(2-methylphenyl)methyl]piperidine
N-(2-hydroxyethyl)-2-(4-methoxyphenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidine
2-{3-[(4aR,8aR)-octahydro-2H-1,4-benzoxazin-4-ylmethyl]phenoxy}acetamide
5-ethyl-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1,3,4-oxadiazol-2-amine
ethyl 1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
N-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
(2S,4R)-4-amino-1-[3-(2,3-dihydro-1H-isoindol-2-yl)benzoyl]-N-ethylpyrrolidine-2-carboxamide
methyl({2-phenylimidazo[1,2-a]pyridin-3-yl}methyl)[1-(pyridin-2-yl)ethyl]amine
4-(furan-2-carbonyl)-N-(2,4,6-trimethylpyridin-3-yl)piperazine-1-carboxamide
N-(1-ethyl-1H-1,2,4-triazol-5-yl)-3-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)benzamide
[(3R,4R)-1-(3-fluorobenzoyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol