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(4aS,8aS)-2-[(2,3-difluoro-6-methoxyphenyl)methyl]-decahydroisoquinolin-4a-ol
1-[3-(2-ethylphenoxy)azetidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
2-[3-(furan-2-yl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-indazol-3-yl)acetamide
N-benzyl-3-[(1S,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N-methylpropanamide
N-methyl-N-[2-(phenylsulfanyl)ethyl]-1,3-benzothiazole-6-carboxamide
2-[4-(1,3-benzoxazol-2-yl)-1H-pyrazol-1-yl]-N-(1,3-dimethyl-1H-pyrazol-5-yl)acetamide
2-(4-methoxyphenyl)-1-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)ethan-1-one
methyl 4-[4-(3-methoxypyrazin-2-yl)piperazin-1-yl]benzoate
N-[1-(2,5-difluorophenyl)cyclopropyl]-1-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine
(3S,4S)-1-(butane-1-sulfonyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
1-[1-(difluoromethyl)-1H-pyrazole-5-carbonyl]-4-(2-methoxyphenoxy)piperidine
2-(2,5-dioxoimidazolidin-1-yl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)acetamide
2-(1,3-dimethyl-4-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}-1H-pyrazolo[3,4-d]pyrimidin-6-yl)pyridine
6-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
3-[1-methyl-3-(pyridin-3-yl)-1H-pyrazol-5-yl]-1-{2-[4-(propan-2-yl)-1,3-thiazol-2-yl]ethyl}urea
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methylacetamide
2-[4-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]-1-(pyrrolidin-1-yl)ethan-1-one
3-{[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}azepan-2-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(pyridin-4-yl)acetamide
N-[1-(2,5-difluorophenyl)cyclopropyl]-6-(methoxymethyl)pyridine-2-carboxamide
3-(dimethylsulfamoyl)-N-methyl-5-[(3-phenylbutyl)amino]-N-[1-(pyridin-2-yl)ethyl]benzamide
1-{1-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]piperidin-4-yl}piperidin-4-ol
(3R,5S)-N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
3-hydroxy-S-{2-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}butane-1-sulfonamido
(4aS,8aR)-6-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
N-cyclopentyl-N-({3-[(4-fluorophenyl)methoxy]phenyl}methyl)-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
3-{2,7-diazaspiro[4.5]decane-7-carbonyl}-1-ethyl-4,6-dimethyl-1,2-dihydropyridin-2-one
methyl 6-benzoyl-2-[(3,4-difluorophenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)cyclohex-1-ene-1-carboxamide
4,4-difluoro-1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
8-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N-cyclohexyl-3-{[4-(4H-1,2,4-triazol-4-yl)phenyl]formamido}propanamide
ethyl 4-{[(2-methylquinolin-5-yl)carbamoyl]amino}piperidine-1-carboxylate
(3S,4R)-4-(3-methoxyphenyl)-1-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)pyrrolidine-3-carboxylic acid
N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-benzyl-9-[(5-fluoro-2-methoxyphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(1,4-oxazepan-4-yl)-4-phenylbutane-1,2-dione
7-[2-(4-fluorobenzenesulfonyl)ethyl]-2-oxa-7-azaspiro[4.5]decan-8-one
1-(4-{2-[4-(2-hydroxyethyl)-1,4-diazepan-1-yl]-2-oxoethoxy}phenyl)propan-1-one
1-(cyclopropylmethyl)-N-ethyl-5-(9H-fluoren-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl](1H-indol-7-ylmethyl)methylamine
3-benzyl-5-(2-ethyl-4-methyl-1,3-oxazol-5-yl)-1H-1,2,4-triazole
6-(4-chlorophenyl)-N-ethyl-N-(2-methylprop-2-en-1-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-ethyl-3-(4-hydroxyphenyl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
(2R,6S)-4-{1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-4-yl}-2,6-dimethylmorpholine
5-(2-fluorophenyl)-N-(thiolan-3-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-(cyclohexylmethyl)-1-cyclopropyl-5-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
{7-[5-(aminomethyl)pyridin-2-yl]-5-methyl-2,3-dihydro-1-benzofuran-2-yl}methanamine