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N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3-fluoro-5-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]benzonitrile
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-2-methylpyrimidine-5-carboxamide
N-ethyl-2-{4-[(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperazin-1-yl}acetamide
4-[(1E)-1-(furan-2-yl)prop-1-en-2-yl]-2-oxo-7-(pyrrolidin-1-yl)-1,2,3,4-tetrahydroquinoline-6-carboxamide
5-methyl-1'-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(2S,4R)-N-ethyl-4-(5-methylthiophene-3-amido)-1-(thiophen-3-ylmethyl)pyrrolidine-2-carboxamide
1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
ethyl 1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylate
2-{3-[3-(7-chloroquinolin-4-yl)phenyl]-1H-pyrazol-1-yl}acetamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(pyridin-2-yl)propanamide
3-(1-{[2-(carboxymethoxy)-5-chlorophenyl]methyl}piperidin-2-yl)propanoic acid
3-[methyl(5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-yl)amino]propan-1-ol
2,3-dimethyl-7-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
4-[3-cyclopropyl-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]-1,2,3-thiadiazole
5-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazin-2-ol
5-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidine-1-carbonyl]pyrazin-2-ol
1-methyl-2-oxo-6-(propan-2-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1,2-dihydropyridine-3-carboxamide
3-(5-{[2-(aminomethyl)morpholin-4-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-3,6-dimethyl-1-benzofuran-2-carboxamide
2-(furan-2-yl)-5-(1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-imidazol-2-yl)pyrimidine
3-(1-{[5-(4-chlorophenyl)furan-2-yl]methyl}azetidin-3-yl)pyridine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-(oxolan-3-yl)-2-pentanoyl-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-[(1-methyl-1H-pyrazol-4-yl)methyl]-decahydro-1,6-naphthyridin-2-one
5-(azepane-1-carbonyl)-N-[(5-chlorothiophen-2-yl)methyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
(2S,4R)-4-hydroxy-N-{[4-(methylsulfanyl)phenyl]methyl}-N-(prop-2-en-1-yl)pyrrolidine-2-carboxamide
2-acetyl-8-(4-ethylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(3R,4S)-4-cyclopropyl-1-[(4,5-dichlorothiophen-2-yl)sulfonyl]pyrrolidin-3-amine
N-methyl-2-(6-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(thiophen-3-ylmethyl)acetamide
5-{3,9-diazaspiro[5.6]dodecane-9-carbonyl}-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2,3,5,6-tetramethylbenzamide
N-[2-(2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamido)ethyl]propanamide
N4-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-6-(propan-2-yl)pyrimidine-2,4-diamine
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-1,1-dioxo-1λ6-thiolane-3-carboxamide
3-{1-[2-(6-oxo-3-phenyl-1,4,5,6-tetrahydropyridazin-1-yl)ethyl]-1H-1,2,3-triazol-4-yl}benzonitrile
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]propan-1-one
1-[3-(2-cyclopropyl-1H-imidazol-1-yl)propyl]-1H-indole
(1R,2R,6S,7S)-4-[(2-methyl-1,3-benzothiazol-6-yl)sulfonyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
4-(cyclopropylmethyl)-1-[2-(3,4-difluorophenyl)acetyl]-1,4-diazepan-5-one
{3-[(4-fluorophenyl)methyl]piperidin-3-yl}methanol
4-[4-({3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenyl]but-3-yn-1-ol
2-(1H-imidazol-1-yl)-1-[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]ethan-1-one
4-(4-ethoxy-3-methylphenyl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-oxobutanamide
2-(2-{3-methyl-1-[(4-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl}ethyl)pyrazine
ethyl 3-[(3-methoxyphenyl)methyl]-1-(2-methyl-1H-1,3-benzodiazole-6-carbonyl)piperidine-3-carboxylate
5-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyrazin-2-ol
4-(4-methyl-1H-pyrazol-1-yl)-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidine-4-carboxylic acid
1-[1-methyl-4-(pyridin-4-ylmethyl)-1,4,9-triazaspiro[5.5]undecan-9-yl]-2-phenoxyethan-1-one
(1S,5R)-6-[(1R,5S,6R)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane