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N-[(2-ethoxyphenyl)methyl]-N-ethyl-2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
1-[(4aR,8aS)-1-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-decahydro-1,6-naphthyridin-6-yl]-2-phenylethan-1-one
2-(naphthalen-1-yl)-5-{[3-(pyridin-4-yl)azetidin-1-yl]methyl}pyrimidine
2-(methylamino)-1-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}ethan-1-one
7-(1-benzothiophen-3-yl)-9-ethoxy-4-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]-N-(3-methylphenyl)propanamide
2-(1-oxo-4-phenyl-1,2-dihydrophthalazin-2-yl)-N-{[7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
5-chloro-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]pyridine-2-carboxamide
3-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-(4-aminopyrimidin-2-yl)-4-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1,4-diazepan-6-ol
1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]-3-(morpholin-4-yl)propan-1-one
N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]propane-1-sulfonamide
3-(2-amino-1,3-thiazol-4-yl)-1-[(3S)-3-(dimethylamino)azepan-1-yl]propan-1-one
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(quinoxaline-6-carbonyl)pyrrolidin-3-yl]methanol
9-methyl-3-(quinoline-6-carbonyl)-3,9-diazaspiro[5.6]dodecane
1-(1H-pyrrole-2-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
3-cyclopropyl-4-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl]-1H-pyrazole
3-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine-3-carbonyl)-4H-pyrido[1,2-a]pyrimidin-4-one
1-{2-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-benzyl-4-methanesulfonyl-1-(3-phenylphenyl)piperazin-2-one
1-[4-(propylsulfanyl)phenyl]-3-[2-(pyrazin-2-yl)ethyl]urea
4-{5-[1-(thiophene-2-carbonyl)pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
(4aS,8aS)-2-[5-(propan-2-yl)pyrimidin-4-yl]-decahydro-2,7-naphthyridin-4a-ol
1-methyl-4-({5-[3-(1H-pyrazol-1-yl)propyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-3-yl}methyl)piperidine
1-[(2,2-dimethyloxan-4-yl)methyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
1-[2-(4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}phenoxy)ethyl]-1H-imidazole
2-cyclopropyl-8-(1,7-dimethyl-1H-indole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[({5-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
[(2-chloro-6-fluoro-3-methylphenyl)methyl](1H-imidazol-2-ylmethyl)methylamine
1-{5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperidin-3-ol
3-{5-[3-(2-methyl-1H-imidazol-1-yl)propyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
1-[5-(1H-indol-5-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]butan-2-ol
3-(diphenylmethyl)-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1,2-oxazole-5-carboxamide
(2S,4S)-N-ethyl-4-(furan-2-amido)-1-[2-(pyridin-4-yl)acetyl]pyrrolidine-2-carboxamide
8-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
ethyl 3-{[2-(cyclohexylmethyl)morpholine-4-carbonyl]amino}propanoate
1-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]-4-phenoxybutan-1-one
3,5-difluoro-N-methyl-N-(quinoxalin-2-ylmethyl)pyridine-2-carboxamide
(2S)-1-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-ethyl-5-({2-[(3-methylpyridin-4-yl)amino]ethyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
3-[8-(2,3-dihydro-1-benzofuran-5-carbonyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl]propanoic acid
N-ethyl-5-[(4-ethylpiperazin-1-yl)methyl]-N-[(2-methylphenyl)methyl]-1,2-oxazole-3-carboxamide
4-ethyl-2-methyl-6-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrimidine
2-(dimethylamino)-2-(4-fluorophenyl)-N-methyl-N-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)acetamide
4-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidine-1-carbonyl]-2-methylphenol
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methyl-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
2-(4-{[cyclohexyl(methyl)amino]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
1-(1H-1,3-benzodiazole-5-carbonyl)-4-[(2-chlorophenyl)methyl]piperidine-4-carboxylic acid
2-[3-(1-methyl-1H-pyrazol-3-yl)phenyl]pyridine
1-[3-(azepane-1-carbonyl)phenyl]-3-[(3-propyl-1,2-oxazol-5-yl)methyl]urea