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2-phenyl-1-[1-(5-propyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]ethan-1-ol
N-(1-{1-[2-(2H-indazol-2-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2,2-dimethylpropanamide
N,N-dimethyl-5-{[4-(quinazolin-4-yl)piperazin-1-yl]methyl}-1,3-thiazol-2-amine
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N,5-dimethyl-2-phenyl-1H-imidazole-4-carboxamide
N-(4-{[2-(3-fluorophenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}phenyl)acetamide
4-(3,6-dimethylpyrazin-2-yl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[2-({2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)ethyl]methanesulfonamide
3-[1-(pentan-2-yl)-1H-pyrazol-5-yl]-1-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}urea
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-3-(1H-pyrazol-1-yl)benzamide
2-[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-3,4-dihydroquinazolin-4-one
N-(furan-3-ylmethyl)-N,2-dimethyl-1H-1,3-benzodiazole-5-carboxamide
8-(2-hydroxy-4-methoxybenzoyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-{5-[5-(propan-2-yl)-1,2-oxazol-3-yl]-1,2,4-oxadiazol-3-yl}pyridine
{[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}(prop-2-en-1-yl)(prop-2-yn-1-yl)amine
N-cyclopropyl-2-(ethylamino)-N-{[4-(methylsulfanyl)phenyl]methyl}pyrimidine-5-carboxamide
1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
7-(3-methylbut-2-enoyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
6-{methyl[2-(pyrrolidin-1-yl)ethyl]amino}pyridine-3-carboxamide
N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-(quinolin-6-yl)pyridine-3-carboxamide
3-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-1-(3-hydroxypropyl)-1-(thiophen-2-ylmethyl)urea
(3S,4S)-1-[2-(morpholin-4-yl)ethyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
(3aS,7aR)-5-methyl-2-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
N-cyclopropyl-4-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}piperazine-2-carboxamide
{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}(methyl){[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
4-chloro-2-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenol
N-{[5-methyl-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}oxolane-3-carboxamide
methyl (1R,3S,3aR,6aS)-5-methyl-1-(2-methylpropyl)-4,6-dioxo-3-[3-(propan-2-yl)-1,2-oxazol-5-yl]-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N'-(4-methylphenyl)-N-[3-(pyridin-3-yl)propyl]propanediamide
4-{[4-(3-ethyl-1,2,4-oxadiazol-5-yl)furan-2-yl]methyl}morpholine
3-(1-methyl-1H-pyrazol-4-yl)-N-[2-(2-methylphenyl)-2-(4-methylpiperidin-1-yl)ethyl]propanamide
methyl 4-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylate
1-{1-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]piperidin-4-yl}pyrrolidin-2-one
(1H-indol-3-ylmethyl)[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]propanamide
2-phenyl-4-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}morpholine
4-methylphenyl (7S,9aR)-6,9-dioxo-7-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
(1R,5R)-6-benzyl-3-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-6-[(2R,5S)-2,5-dimethylpyrrolidine-1-carbonyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-(3,4-dimethylphenoxymethyl)-1,2-oxazole-3-carboxamide
1-(3,5-dimethylphenyl)-N-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
3-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-methyl-1-[3-(trifluoromethoxy)phenyl]urea
9-[2-(4-chlorophenyl)-2-hydroxyacetyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
(3R,4R)-1-(1-cyclobutanecarbonylpiperidin-4-yl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
(1R,5S,6S)-N-[1-benzyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(5-methylthiophen-2-yl)methyl]amine
7-methyl-2-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
4-[(cyclopropylmethyl)sulfamoyl]-N-[2-(1H-pyrrol-1-yl)ethyl]benzamide
4-[1-(2-methoxyethyl)-5-oxopyrrolidine-3-carbonyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
(2S,4S)-4-amino-1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-N-methylpyrrolidine-2-carboxamide
N-({1-[(4,6-dimethylpyrimidin-2-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)-N-methylacetamide