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1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
3-{[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]amino}-N-(1,3-thiazol-2-yl)propanamide
{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}[(4-phenyl-1,3-thiazol-5-yl)methyl]amine
1-methyl-4-({5-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1,2,4-oxadiazol-3-yl}methyl)piperidine
2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[3-(oxolan-3-yl)propyl]-1,3-oxazole-4-carboxamide
2-[3-(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)phenoxy]acetamide
3-[2-(dimethylamino)ethyl]-8-(1-methoxypropan-2-yl)-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{2-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propanamido]ethyl}piperidine-3-carboxamide
3-({2-methyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}methyl)benzonitrile
4-benzyl-1-[(1-benzyl-1H-imidazol-5-yl)methyl]pyrrolidin-2-one
6-oxo-N-[2-(pyridin-3-yloxy)phenyl]piperazine-2-carboxamide
4-{2-methyl-2-[1-methyl-3-(pyridin-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]propyl}morpholine
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-1H-pyrazole-3-carboxamide
5-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]-1,2-dihydropyridin-2-one
[(3R,4R)-4-[(dimethylamino)methyl]-1-(4-methanesulfonylbenzoyl)pyrrolidin-3-yl]methanol
1-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-4-methylpiperazine
2-[5-(3,6-dimethyl-1-benzofuran-2-yl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
N-[(2,6-difluoro-3-methylphenyl)methyl]-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-methoxy-N-{[8-methyl-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}benzene-1-sulfonamide
2-(furan-2-yl)-N-methyl-2-oxo-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}acetamide
1-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}ethan-1-one
1-(3-ethylpiperazin-1-yl)-3-(4-methylbenzenesulfonyl)propan-1-one
1-[(3,4-dimethylphenyl)methyl]-2-oxo-3-[2-(pyridin-2-yl)ethyl]-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
2-chloro-N-(2-{[1-(propan-2-yl)-1H-pyrazol-4-yl]formamido}ethyl)benzamide
2-cyclohexyl-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1,3-benzoxazole-6-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-5-[(dimethyl-1,3-thiazol-5-yl)methyl]-1H-1,2,4-triazole
1-[(3,5-difluorophenyl)methyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
[2-({4-[(5-methylthiophen-2-yl)methyl]piperazin-1-yl}methyl)phenyl]methanol
N-(1-{1-[3-(2-chlorophenyl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
2-(1-cyclopentyl-4-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-2-yl)ethan-1-ol
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-N-ethyl-N-(2-methylprop-2-en-1-yl)propanamide
{4-[(3-methoxyphenyl)methyl]-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}methanol
methyl 4-[4-phenyl-5-(1-propyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]butanoate
(3R,5R)-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
(4aS,8aR)-6-[2-(5-amino-1,3,4-thiadiazol-2-yl)acetyl]-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
4-[(2-hydroxyethyl)sulfamoyl]-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]benzamide
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(1,3-thiazol-2-yl)piperidine
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
(1-methyl-1H-imidazol-2-yl)[1-(3-phenyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]methanol
3-(5-amino-1H-1,2,4-triazol-3-yl)-N-[(1S,2R)-2-[(1-propylpiperidin-4-yl)amino]cyclobutyl]propanamide
8-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(3-methylbutyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
9-(5-chloropyridin-2-yl)-2-(cyclopropylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}pyrrolidin-2-yl)pyridine
1-[(1R,3S,5S)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octan-8-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
3-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-2-methylphenol
(2S,4R)-N-methyl-1-[(6-methylpyridin-2-yl)methyl]-4-[2-(thiophen-2-yl)acetamido]pyrrolidine-2-carboxamide
2-[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]-1-(oxan-4-ylmethyl)-1H-imidazole
1-{2-[4-(2-methoxyethoxy)phenyl]pyrimidin-4-yl}pyrrolidin-3-ol
1-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-1-methyl-3-[2-methyl-3-(pyrrolidin-1-yl)phenyl]urea
1-methyl-3-propyl-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazole-5-carboxamide