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2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(pyrrolidine-1-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
4-(4-methyl-1H-pyrazol-1-yl)thiophene-2-carboxamide
(2-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)urea
[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl](methyl)[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amine
(1S,4S)-2-(3,5-dichloro-4-methylbenzoyl)-2,5-diazabicyclo[2.2.1]heptane
(3S)-4-{[3-(cyclopentyloxy)phenyl]methyl}-3-ethylmorpholine
2-chloro-N-(1-{1-[(methylcarbamoyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
4-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-1-propylpiperidine
2-amino-6-{4-[2-methyl-2-(morpholin-4-yl)propyl]piperazin-1-yl}pyrimidin-4-ol
4-benzyl-N-(2-fluoro-4-methoxyphenyl)-4-hydroxypiperidine-1-carboxamide
4-methoxy-6-(3-{1-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
2-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
5-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-2-ethyl-4-methyl-1,3-thiazole
2-[2-(dimethylamino)ethyl]-9-(4-hydroxy-3-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(4-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}piperazin-1-yl)pyridine-3-carbonitrile
N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)propanamide
4-{4-[1-(4-methoxyphenyl)cyclopentanecarbonyl]piperazin-1-yl}-2-(pyridin-4-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
(1S,5R)-3-(2,1,3-benzothiadiazol-5-ylmethyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3R,4S)-4-propyl-1-(3,5,7-trimethyl-1H-indole-2-carbonyl)pyrrolidin-3-amine
1-[4-(3-{[(cyclohex-3-en-1-ylmethyl)amino]methyl}pyridin-2-yl)piperazin-1-yl]ethan-1-one
[(3R,4R)-1-(2,3-difluoro-4-methoxybenzoyl)-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-7-[(thiophen-2-ylmethyl)amino]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-5-methylpyrazine
1-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-4-(2-methoxyphenoxy)piperidine
N-methyl-N-[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(pyridazine-4-carbonyl)piperidine-4-carboxamide
1-cyclopropyl-N-{[1-(4-fluorophenyl)cyclopentyl]methyl}-5-oxopyrrolidine-3-carboxamide
2-methyl-6-[4-(4-methylphenoxy)piperidine-1-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
2-(2-aminoethyl)-N-ethyl-N-(oxan-2-ylmethyl)quinazolin-4-amine
5-methyl-1'-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-[3-(furan-2-yl)-5-[1-(pyridin-2-yl)piperidin-3-yl]-1H-1,2,4-triazol-1-yl]acetic acid
(3S,4R)-1-(propane-1-sulfonyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-7-hydroxy-6-methyl-1,2,3,4-tetrahydroquinolin-2-one
1-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-(3-methylpyridin-4-yl)-1,4-diazepane
methyl 3-[3-(cyclopropylcarbamoyl)-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanoate
3-{[(3S,4S)-3,4-bis(hydroxymethyl)pyrrolidin-1-yl]methyl}-6-ethoxy-1,2-dihydroquinolin-2-one
N-[2-(5-methylthiophen-2-yl)ethyl]-1,1-dioxo-3,4-dihydro-2H-1λ6,2-benzothiazine-3-carboxamide
N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
3-({3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}methyl)-1λ6-thiane-1,1-dione
dimethyl({4-[1-(pyridine-4-carbonyl)piperidin-2-yl]phenyl}methyl)amine
2-[(2S)-2-aminopentanoyl]-N-[(5-methylfuran-2-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
2-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(4-chlorophenoxy)-N-(oxan-4-ylmethyl)piperidine-4-carboxamide
5-[1-(2,3-dihydro-1H-inden-4-yl)-3-methyl-1H-1,2,4-triazol-5-yl]-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[5-(2-amino-4-methyl-1,3-benzothiazole-6-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
1-[4-(methylamino)pyrimidin-2-yl]-4-(1H-1,2,3-triazol-4-ylmethyl)-1,4-diazepane-6-carboxylic acid
4-[(4-fluorophenyl)methyl]-1-[(2-methoxyphenyl)methyl]-1,4-diazepan-5-one
methyl 3-[(5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-1H-pyrazol-4-yl)formamido]propanoate
1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-6-methyl-4-(trifluoromethyl)-1,2-dihydropyridin-2-one