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N-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]benzamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-5-[(dimethylamino)methyl]phenol
3-(1-cyclopentylpiperidin-3-yl)-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(5-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
2-methyl-6-[1-(2-phenylethyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-2,3-dihydropyridazin-3-one
3-[(5-amino-1,3,4-thiadiazol-2-yl)methyl]-1-[4-(oxan-2-ylmethoxy)phenyl]urea
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-2-(ethylamino)pyrimidine-5-carboxamide
7-fluoro-N-methyl-2-oxo-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1,2-dihydroquinoline-4-carboxamide
6-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-8-yl]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
2,2-dimethyl-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
1-{4-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]phenyl}ethan-1-one
[(3R,4R)-4-(azepan-1-ylmethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl]methanol
3-(3-methylbut-2-en-1-yl)-1-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxylic acid
{4-[(2-cyclohexylpyrimidin-5-yl)methyl]morpholin-3-yl}methanol
3-[5-(4-propylpyrimidine-5-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
N-[3-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-methyl-3-[methyl({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl})amino]propanamide
2-(3-methoxypropyl)-8-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
6-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carboxylic acid
3-{4-[(2-phenylpyrimidin-5-yl)methyl]piperazin-1-yl}-1λ6-thiolane-1,1-dione
3-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-oxo-3,4-dihydrophthalazine-1-carboxamide
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-(2-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}-1H-pyrrol-1-yl)pyridine
1-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propane-1,2-dione
4-[2-(2-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]thiomorpholine
N-[(4-chlorophenyl)(phenyl)methyl]-2-ethyl-6-methyl-4-oxo-1-[2-(piperidin-1-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
2-ethoxy-N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-phenylpyrrolidin-3-yl]acetamide
N-methyl-N-{2-phenyl-1-[1-(quinoxaline-6-carbonyl)piperidin-4-yl]ethyl}thiophene-2-carboxamide
2-(1-cyclohexyl-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl)ethan-1-ol
3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]propanamide
3-(2-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-2-oxoethyl)-1,2,3-oxadiazol-3-ium-5-olate
4-(4-methylpiperazin-1-yl)-6-{1H-pyrazolo[3,4-b]pyridin-1-yl}quinazoline
diphenyl({1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl})methanol
2-(4-fluorophenyl)-4-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}morpholine
1,5-dimethyl-2-phenyl-4-{[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-2,3-dihydro-1H-pyrazol-3-one
4-cyano-N-[(3R,4S)-4-propyl-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]oxane-4-carboxamide
N-methyl-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
N-methyl-3-[(2R)-2-methylpiperazine-1-carbonyl]-N-[2-(1H-pyrazol-1-yl)ethyl]benzene-1-sulfonamide
4-methoxy-N-[(3-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)cyclohexane-1-carboxamide
N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-N,2-dimethyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
5-{1-[(2,5-difluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
3-{2-oxo-2-[2-(pyridin-3-yl)piperidin-1-yl]ethyl}-3,4-dihydroquinazolin-4-one
(4aR,8aR)-2-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
N-[4-(4-fluoro-2-methoxyphenyl)phenyl]-2-methoxyacetamide
3-{1-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]piperidin-4-yl}phenol
6-{3-[(4-methoxyphenyl)methyl]-1-methyl-1H-1,2,4-triazol-5-yl}-1,2,3,4-tetrahydroquinoxaline-2,3-dione
N-[4-(4-fluorophenoxy)phenyl]-3-methoxypiperidine-1-carboxamide
N-benzyl-1-(2-hydroxyethyl)-5-(quinolin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-2-(2H-1,3-benzodioxol-5-yl)ethan-1-one