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N3-methyl-4-oxo-1-(3-phenylpropyl)-N5-(2,2,2-trifluoroethyl)-1,4-dihydropyridine-3,5-dicarboxamide
4-(pyridin-3-yl)-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]pyrimidin-2-amine
1-methyl-4-{3-[5-(pentan-2-yl)-4-phenyl-1H-imidazol-1-yl]propoxy}piperidine
4-[(4-fluorophenyl)methyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine
2-{5-[3-(1H-imidazol-1-yl)propyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
3-(4-methanesulfonyl-2-oxopiperazin-1-yl)benzonitrile
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carboxamide
1-[(2,6-difluorophenyl)methyl]-3-[3-(dimethylamino)propyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
N-(1-cyclopropylethyl)-2-[1-(4-methoxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
4-({[1-(2-methoxyethyl)piperidin-3-yl]methyl}(methyl)amino)-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-6-(4-methyl-1,4-diazepane-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-(2-{1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidin-2-yl}ethyl)acetamide
5-[1-(2,2-dimethylpropanoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-(5-acetyl-2-ethoxyphenyl)-3-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]urea
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-hydroxy-2-methylpropanamide
methyl({[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl})(quinolin-2-ylmethyl)amine
3-(5-chloro-1-methyl-4-{[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methyl}-1H-pyrazol-3-yl)-5-methyl-1,2-oxazole
N-[(2-chloro-6-fluorophenyl)methyl]-N-ethyl-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
methyl 2-[(4-chlorophenyl)sulfamoyl]-6-(3,3-dimethylbutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-methyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-4-oxo-3,4-dihydroquinazoline-2-carboxamide
N-{2-[4-(4-chlorophenyl)-4H-1,2,4-triazol-3-yl]ethyl}aniline
(benzylsulfamoyl)[2-(4-methylpiperazin-1-yl)butyl]amine
1-(4-methoxyphenyl)-4-[1-(3-phenylpropyl)piperidin-3-yl]piperazine
2-(ethoxymethyl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-ethyl-8-{4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzoyl}-2,8-diazaspiro[4.5]decan-3-one
3-(3-methoxybenzoyl)-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine
4-[2-(3-methylbutoxy)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
4-({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)-1-(2-methoxyethyl)pyrrolidin-2-one
5-[methyl(2-phenylethyl)amino]-2-[2-(1H-pyrazol-1-yl)ethyl]-2,3-dihydropyridazin-3-one
1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
3,3-dimethyl-1-[(5-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]urea
1-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(methylsulfanyl)propan-1-one
4-(2-methylquinolin-6-yl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-4-ol
2-(2H-1,3-benzodioxol-5-yl)-4-{1-[(6-chloropyridin-3-yl)methyl]pyrrolidin-3-yl}pyridine
3-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]phenol
2-(3-methylbut-2-en-1-yl)-8-[2-(trimethyl-1H-pyrazol-1-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
2-(2-methoxyethyl)-8-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
4-(4-{[4-(4-methylphenyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)pyrimidin-2-amine
N-(4-methoxy-2-methylphenyl)-3-[1-(1H-pyrrole-2-carbonyl)piperidin-3-yl]propanamide
(2S,4R)-4-amino-1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-(4-fluorophenyl)-1-(quinoxalin-2-yl)piperidin-3-amine
2-methoxy-1-{1'-[2-(pyridin-2-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
methyl N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)carbamate
1-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-2-cyclopropyl-1H-imidazole
4,6-dimethyl-2-{4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperazin-1-yl}pyrimidine
6-methoxy-N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-{3-[(3S,4S)-4-(4-fluorophenyl)-3-hydroxypiperidine-1-carbonyl]phenyl}imidazolidin-2-one
5-methyl-3-(2,2,6,6-tetramethylpiperidin-4-yl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
benzyl({[3-(3-ethyl-4-methylpiperazine-1-carbonyl)-1,2-oxazol-5-yl]methyl})methylamine
7-(2-hydroxyethyl)-2-({2-methyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)-2,7-diazaspiro[4.5]decan-6-one