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2-[4-(1,4-diazepan-1-ylmethyl)phenyl]-6-(4-fluorophenyl)-3,4-dihydropyrimidin-4-one
1-methyl-1-[2-(pyridin-2-yl)ethyl]-3-(5,7,8-trimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea
2-(3-methylphenyl)-5-{[3-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]methyl}pyrimidine
(2R)-2-(methoxymethyl)-1-[5-(methoxymethyl)furan-2-carbonyl]pyrrolidine
1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-3-methoxy-1,2-dihydropyridin-2-one
5,6-dimethyl-2-oxo-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)-1,2-dihydropyridine-3-carboxamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-3-(2-oxopyrrolidin-1-yl)benzamide
1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(methoxymethyl)-N-[(4-phenyloxan-4-yl)methyl]-1H-pyrazole-4-carboxamide
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-(3-phenylpropyl)piperidin-3-amine
N-[4-methoxy-2-(2-methylpropanamido)phenyl]-3-oxo-2,3-dihydro-1H-indene-1-carboxamide
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(pyridin-3-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-{1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}thiomorpholine
2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
dimethyl(2-{2-[1-(5-methylpyridin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
(5-{1-[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]-1H-imidazol-2-yl}furan-2-yl)methanol
4-[5-({[2-(azepan-1-yl)ethyl](ethyl)amino}methyl)thiophen-2-yl]-2-methylbut-3-yn-2-ol
2-({2-[1-(pyrrolidine-1-sulfonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[(2R,3R)-2-methoxy-1'-[2-(1H-1,2,4-triazol-1-yl)acetyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
N-[(2S,4R,6S)-2-benzyl-6-(pyridin-3-yl)oxan-4-yl]benzamide
N-{[7-methoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-5-methyl-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
(4aS,7aR)-1-[(3-ethoxyphenyl)methyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-tert-butyl-5-[4-(pyridin-4-yloxy)piperidine-1-carbonyl]pyrimidin-4-ol
5-({3-[(4aS,8aR)-decahydroisoquinoline-2-carbonyl]-1,2-oxazol-5-yl}methoxy)isoquinoline
1-(2-chloroprop-2-en-1-yl)-3-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}methyl)-7-fluoro-1,2-dihydroquinolin-2-one
(1R,5R)-3-[2-(difluoromethoxy)benzoyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonane
ethyl 1-(2-hydroxyethyl)-5-(naphthalen-1-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-cyclopropyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
2-(2,2-diphenylethyl)-4-(1H-imidazol-2-ylmethyl)morpholine
4-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
dimethyl[3-(3-{[(1S,6R)-3-methyl-3,9-diazabicyclo[4.2.1]nonan-9-yl]methyl}phenoxy)propyl]amine
2-[5-(1H-imidazol-4-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]-1-(prop-2-en-1-yl)-1H-1,3-benzodiazole
1-[3-(morpholin-4-yl)propyl]-6-oxo-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidine-3-carboxamide
1-(5-ethyl-1,3,4-oxadiazol-2-yl)-4-methanesulfonylpiperazine
1-{3-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-4-(thiophen-2-yl)butan-1-one
2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]acetamide
N-[(2E)-but-2-en-1-yl]-N-(butan-2-yl)-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
3-(2-oxo-2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-2,3-dihydro-1H-isoindol-1-one
5-amino-3-(3-methyl-1,2-benzoxazol-5-yl)-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}-1-(1,3-thiazole-5-carbonyl)piperidine
1-ethyl-4-({9-ethyl-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}methyl)-1H-pyrrole-2-carbonitrile
3-(2H-1,3-benzodioxol-5-yl)-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}propanamide
2-{1-[4-(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,3-triazol-1-yl]propyl}-3-methylpyridine
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(pyrimidin-2-ylsulfanyl)acetamide
2-[5-(butoxymethyl)-3-phenyl-1H-1,2,4-triazol-1-yl]pyridine
3-{4-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}benzonitrile
2-(3-methyl-5-{[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]methyl}-1H-1,2,4-triazol-1-yl)benzoic acid
N-[3-(N-methylacetamido)phenyl]-4-(1-methylpiperidin-4-yl)piperazine-1-carboxamide
2-[2-fluoro-6-(propan-2-yloxy)phenyl]-2-[4-(pyridin-4-yl)piperidin-1-yl]acetic acid
1-[(4-methoxyphenyl)methyl]-4-(2-methylfuran-3-carbonyl)piperazin-2-one
1-(3,5-dimethyl-1-benzofuran-2-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol