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(3aR,7aS)-2-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)cyclopropane-1-carboxamide
(3aS,6aR)-3-[2-(4-fluorophenyl)ethyl]-2-oxo-N-(propan-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carboxamide
4-{4-[(3ar,6ar)-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]piperazin-1-yl}benzonitrile
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(pyridin-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-5-methoxy-1-methyl-1H-indole-2-carboxamide
5-fluoro-2-[1-(5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
(2S)-2-amino-N-[(5-methylthiophen-2-yl)methyl]-N-(prop-2-en-1-yl)-3-(1,3-thiazol-4-yl)propanamide
N-(3-{2-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]-2-oxoethoxy}phenyl)propanamide
N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-1H-imidazole-5-carboxamide
N,N-diethyl-2-(methoxymethyl)-6-methyl-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3-carboxamide
N-methyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-(oxan-4-yl)-1,2-oxazole-3-carboxamide
2-tert-butyl-7,7-dimethyl-N-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-5,6,7,8-tetrahydroquinazolin-5-amine
3-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(trifluoromethyl)phenyl]urea
{2-[1-(3-chlorophenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]ethyl}dimethylamine
1-{2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzoyl}piperidin-3-ol
8-(dimethyl-1,3-thiazole-5-carbonyl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-2-(pyrimidin-2-ylsulfanyl)acetamide
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
N-[1-(thiophen-2-yl)propan-2-yl]-1-(4,6,7-trimethylquinazolin-2-yl)piperidin-4-amine
3-[2-(2-fluorophenyl)ethyl]-1-(4-methyl-1H-imidazole-5-carbonyl)piperidine
(2S,4R)-4-amino-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-[4-(naphthalen-2-yl)piperazin-1-yl]propan-1-one
N-cyclohexyl-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
5-(4-fluorophenyl)-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-tert-butyl-1-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}urea
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidine
(2R,6R)-4-{2-[(dimethylcarbamoyl)amino]acetyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(dimethyl-1,2-oxazole-4-carbonyl)piperidine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{[2-(ethylamino)pyrimidin-5-yl]methyl}piperidin-3-ol
6-methyl-2-[4-({methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
1-[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl]butane-1,2-dione
4,5,6-trimethyl-3-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1,2-dihydropyridin-2-one
5-cyclopropyl-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]methanol
7-methyl-2-{6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
2-(naphthalen-1-yl)-2-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]acetic acid
1-(1-hydroxycyclohexanecarbonyl)-1,4-diazepane-6-carboxylic acid
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(pyridazine-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzamide
2-methyl-4-propyl-6-[4-(pyrimidin-5-ylmethyl)piperazin-1-yl]pyrimidine
1-(oxolan-3-ylmethyl)-5,5-diphenylpiperidin-2-one
1-ethyl-5-(2-phenyl-1H-imidazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-(3-methanesulfonamidophenyl)-3-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}urea
4-[2-(adamantan-1-yl)acetamido]-N-ethylpiperidine-1-carboxamide
N-[(2S)-butan-2-yl]-2-[2-(dimethylamino)pyrimidin-5-yl]-8-methylquinoline-4-carboxamide
3-(tert-butylsulfamoyl)-5-[(furan-3-ylmethyl)amino]-N-[(1-methylpiperidin-3-yl)methyl]benzamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-3-(1-methyl-1H-pyrazol-4-yl)propanamide
4-{5-methyl-4-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-2-oxopiperazin-1-yl}benzonitrile
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-1-[3-(methylsulfanyl)propyl]pyrrolidine-2-carboxamide