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2,6-dimethyl-N-[2-(1H-1,2,4-triazol-1-yl)propyl]quinoline-3-carboxamide
1-(1-ethylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
1-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-[6-(morpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazine-1-carbaldehyde
3-hydroxy-1-(6-hydroxy-4-{thieno[2,3-d]pyrimidin-4-yl}-1,4-diazepan-1-yl)propan-1-one
4-(5,6-dimethylpyridine-3-carbonyl)-3-ethylpiperazin-2-one
[1-(6-methylpyridazin-3-yl)-3-(3-phenylpropyl)piperidin-3-yl]methanol
2-(3-fluorophenyl)-4-[1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]pyridine
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-1-(5,6,7,8-tetrahydro-1,6-naphthyridin-6-yl)propan-1-one
8-[5-(pyrrolidine-1-carbonyl)pyridin-2-yl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
7-[(3-methylphenyl)methyl]-2-(6-oxo-1,6-dihydropyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-(1,1-dioxo-1λ6-thian-4-yl)-N-methyl-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
3-(1H-1,3-benzodiazol-2-yl)-N-butyl-N-[(3-methoxyphenyl)methyl]propanamide
8-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2S,4R)-N,N-diethyl-4-(2-hydroxyacetamido)-1-[2-(4-hydroxyphenyl)acetyl]pyrrolidine-2-carboxamide
N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
2-chloro-3-{[(1-hydroxybutan-2-yl)(thiophen-2-ylmethyl)amino]methyl}-6-methoxyphenol
2-{[2-(6-chloro-2-fluoro-3-methoxyphenyl)-1H-imidazol-1-yl]methyl}-5-methylpyrazine
4-(1-{1-[(3,4-dimethylphenyl)methyl]piperidin-4-yl}ethyl)morpholine
8-methoxy-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
{1-[3-(methylsulfanyl)propyl]-3-(2-phenylethyl)piperidin-3-yl}methanol
2-{2-[(3-ethyl-4-methylpiperazin-1-yl)methyl]-4-(pyrimidin-2-yl)phenoxy}acetic acid
1-(morpholin-4-yl)-3-[5-(pent-2-yn-1-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propan-1-one
N-methyl-3-(thiophen-2-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[1-(thiophen-2-yl)ethyl]amine
2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-(thiomorpholin-4-yl)ethan-1-one
benzyl N-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]carbamate
N-cyclopropyl-4-(3-fluoropyridin-4-yl)piperazine-2-carboxamide
2-{[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]methyl}benzoic acid
2-(3,4-dimethoxyphenyl)-1-[1-(2,2-dimethyloxane-4-carbonyl)piperidin-4-yl]-5-fluoro-1H-1,3-benzodiazole
{3-[(2,4-difluorophenyl)methyl]-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-3-yl}methanol
(1S,3R)-3-amino-N-(1H-1,2,3-benzotriazol-4-yl)cyclopentane-1-carboxamide
2,8-dimethyl-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}quinoline-4-carboxamide
4-ethyl-1-[2-(4-methylphenyl)quinoline-4-carbonyl]-1,4-diazepan-5-one
1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-oxo-5-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-2,3-dihydro-1H-imidazole-4-carboxylic acid
N-ethyl-N-[2-(4-methylbenzenesulfonyl)ethyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-{2-[5-(hydroxymethyl)furan-2-carbonyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}pyridine-2-carboxamide
1-(3-methyl-4-{[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}phenyl)-1H-pyrazole
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1-methyl-3-(1-propyl-1H-1,3-benzodiazol-5-yl)urea
6-ethyl-1,5-dimethyl-2-oxo-N-(2,2,2-trifluoroethyl)-1,2-dihydropyridine-3-carboxamide
2-methoxy-3-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
1-[4-(2-aminopyrimidin-4-yl)piperidin-1-yl]-2-(pyridin-3-yl)ethane-1,2-dione
2-amino-N-[3-(4-chlorophenyl)propyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-[(1-tert-butyl-5-oxopyrrolidin-3-yl)methyl]-3-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
(3aR,6aR)-2-(5-acetylpyridin-2-yl)-5-cyclopropanecarbonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(4aS,8aR)-1-(3-methoxypropyl)-6-(pyridazine-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-2-(azepan-1-yl)acetamide
N4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
8-fluoro-2-{1-oxa-8-azaspiro[4.6]undecane-8-carbonyl}-1,4-dihydroquinolin-4-one