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1-(4-{[2-(4-fluorophenyl)imidazo[1,2-a]pyridin-3-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
(3aS,6aR)-5-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-3-[3-(4-fluorophenyl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
[(5-{1-benzyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}furan-2-yl)methyl]dimethylamine
3-[5-({2-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}methyl)-1,2,4-oxadiazol-3-yl]pyridine
5-(5-methoxy-1-methyl-1H-indole-2-carbonyl)-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
3-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidine-1-carbonyl]-1-methyl-1,2,5,6,7,8-hexahydroquinolin-2-one
2-(2-hydroxyethyl)-8-[(1-methyl-1H-imidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
(3S,4R)-N,N-dimethyl-4-propyl-1-[2-(trifluoromethyl)benzenesulfonyl]pyrrolidin-3-amine
8-fluoro-2-{[4-(morpholine-4-carbonyl)piperazin-1-yl]methyl}quinolin-4-ol
1-[cyclohexyl(methyl)amino]-3-{3-[(4,4-difluoropiperidin-1-yl)methyl]phenoxy}propan-2-ol
5-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]-2-(methoxymethyl)pyrimidine
(2-methoxyethyl)({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})(1,3-thiazol-2-ylmethyl)amine
4-{4-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridin-6-yl]piperidin-1-yl}-N,N,6-trimethylpyrimidin-2-amine
2-cyclopropyl-5-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidine-1-carbonyl]pyrimidin-4-ol
N2-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-6-(3-fluorophenyl)pyrazine-2,3-diamine
1-(2-ethylpyridine-4-carbonyl)-4-[(3-fluorophenyl)methyl]piperazine
N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}imidazo[1,2-a]pyridine-6-carboxamide
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
2-(2-methoxyphenyl)-4-[(1-methyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-[butyl(methyl)sulfamoyl]-N-[1-(6-methylpyridin-3-yl)ethyl]benzamide
2-(4-propanoylphenoxy)-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]acetamide
2-ethyl-9-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[2-(1H-imidazol-4-yl)ethyl]-9-(6-methylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
N,N-dimethyl-3-{3-[({2-[methyl(phenyl)amino]ethyl}carbamoyl)amino]phenyl}propanamide
1-[(4-fluorophenyl)methyl]-4-(3-methoxypyridine-2-carbonyl)-2-(propan-2-yl)-1,4-diazepane
6-(3-{4-[(3-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-oxopropyl)-2,3-dihydropyridazin-3-one
{4-[(3-fluorophenyl)methyl]-1-(6-methylpyridazin-3-yl)piperidin-4-yl}methanol
4-(3-{[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}propyl)-1,2,5-oxadiazole-3-carboxylic acid
N-methyl-N-[3-(3-methylphenoxy)propyl]-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
[(3R,4S)-4-(morpholin-4-ylmethyl)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]methanol
1-(3-methoxyphenyl)-4-[4-(propan-2-yl)benzoyl]piperazin-2-one
N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
2-[2-(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)-6-methoxyphenoxy]propanoic acid
3-(4-chloro-3-fluorophenyl)-6-(propan-2-yloxy)pyridazine
4-[4-(2-methoxyphenyl)-4H-1,2,4-triazol-3-yl]phenol
N-[2-(4-chlorophenyl)ethyl]-1-[2-(dimethylamino)ethyl]-5-oxopyrrolidine-3-carboxamide
N-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-6-(piperidin-4-yl)pyrimidin-4-amine
1-(5-chloropyridin-2-yl)-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylic acid
9-ethyl-N,1-dimethyl-10-oxo-N-phenyl-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
3-ethoxy-1-[9-hydroxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
1-(3-phenylpropyl)-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-1,4-diazepane
N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
5-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
1-methyl-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
N-(1-{[5-(4-ethyl-5-methylpyrimidin-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}pyrrolidin-3-yl)acetamide
1-[(1-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}piperidin-3-yl)methyl]-1H-1,2,3-triazole-4-carboxylic acid
2,6-difluoro-4-methoxy-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]benzamide
N-({7-[(3-methylthiophen-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-phenoxyacetamide
3-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidine-1-carbonyl]pyridin-2-ol
2-(dimethyl-1,3-thiazol-5-yl)-N-[(4-sulfamoylphenyl)methyl]acetamide