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3-[methyl({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amino]-1-phenylpropan-1-ol
{4-[3-(dimethylamino)benzoyl]-1-methylpiperazin-2-yl}methanol
3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-methyl-1-[2-methyl-5-(4H-1,2,4-triazol-4-yl)phenyl]urea
(3aR,6aS)-N-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-8-yl)-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide
5-(5-methyl-2-phenylfuran-3-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
1-[1'-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
8-[(3-hydroxyphenyl)methyl]-3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-({4-[(2-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-hydroxy-2-(thiophen-2-yl)pyrimidine-5-carboxamide
5-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}-1H-1,2,3-benzotriazole
4-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-carbonyl]-8-methoxy-1,2,3,4-tetrahydroquinolin-2-one
{[4-(difluoromethoxy)phenyl]methyl}(ethyl)(oxan-2-ylmethyl)amine
3-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]-1H-indole
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methyl-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
6-{3-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-2,3-dihydropyridazin-3-one
1-[5-(2-chloro-4-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]azocane
8-fluoro-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]quinoline-2-carboxamide
1-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
4-(3,3-difluoropiperidine-1-carbonyl)-7,8-dimethyl-2-(pyrimidin-5-yl)quinoline
2-(naphthalen-2-yloxy)-1-[3-(pyridin-3-yl)azetidin-1-yl]propan-1-one
4-{4-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
1-[(5-methylfuran-2-yl)methyl]-4-oxo-N-(prop-2-en-1-yl)-5-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl}-1,4-dihydropyridine-3-carboxamide
4-[3-(2-amino-1,3-thiazol-4-yl)propanamido]-N-phenylpiperidine-1-carboxamide
1-[4-({methyl[1-(pyrazin-2-yl)propan-2-yl]amino}methyl)thiophen-2-yl]ethan-1-one
1-(3-{2-[(2-methoxyethyl)sulfanyl]-5-(3-methoxyphenyl)pyrimidin-4-yl}piperidin-1-yl)-2-(1,3-thiazol-4-yl)ethan-1-one
N-[4-(3-fluorophenyl)phenyl]-1-(1H-imidazol-4-ylmethyl)pyrrolidine-2-carboxamide
[4-methyl-5-(1-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methanol
2,3-dimethyl-6-[1-(propan-2-yl)piperidine-4-carbonyl]-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
8-(4-cyclobutyl-6-methylpyrimidin-2-yl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}cyclohex-3-ene-1-carboxamide
N-[(2S)-1-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-4-methyl-1-oxopentan-2-yl]acetamide
3-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N,N-dimethylbenzamide
N-(2-{2-[(2,6-dichlorophenyl)methyl]-6-oxo-1,6-dihydropyrimidin-4-yl}ethyl)acetamide
1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-(5-methanesulfonyl-2-methylphenyl)urea
2-[5-(5-methoxy-1,2-dimethyl-1H-indol-3-yl)-1-methyl-1H-1,2,4-triazol-3-yl]acetamide
N-ethyl-N-methyl-2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,3-oxazole-4-carboxamide
N-(1-carbamoylcycloheptyl)-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
(1-{[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-3-(3-methylbut-2-en-1-yl)piperidin-3-yl)methanol
2-methyl-8-[(2-methyl-1,3-benzothiazol-6-yl)sulfonyl]-2,8-diazaspiro[4.5]decan-3-one
N-[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
3-methyl-4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1-(2-methylpropyl)piperazin-2-one
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2,3,4,9-tetrahydro-1H-carbazole-6-carboxamide
N'-(3-ethylphenyl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}butanediamide
2-{[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}benzoic acid
2-amino-4-(3-ethyl-1H-pyrazol-5-yl)-6-(furan-2-yl)pyridine-3-carbonitrile
3-{[1-(2-hydroxyethyl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
3-[(dimethylamino)methyl]-1-({2-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)pyrrolidin-3-ol
5-{[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]methyl}pyrimidin-2-amine
N-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]phenyl}cyclopropanecarboxamide
N-[(5-carbamoyl-1,2,4-oxadiazol-3-yl)methyl]-2,7,8-trimethylquinoline-4-carboxamide