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methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}amine
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(1H-pyrrole-2-carbonyl)piperidine
4-{1-[6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidine-4-carbonyl}morpholine
N-{1-[1-(2-hydroxypropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-methoxybenzamide
1-[4-(azetidin-1-ylmethyl)-2-methoxyphenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
1-[(5-methylthiophen-2-yl)methyl]-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
2-[4-(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzoyl)piperazin-1-yl]ethan-1-ol
2-[4-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]pyrrolidine-1-carboxamide
methyl 1-methoxy-8-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-(furan-2-yl)-2-oxoacetamide
N-(1-benzylpiperidin-4-yl)-2-(cyclopentylmethyl)-1,6-dimethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-ethyl-3-methylpiperazin-2-one
2-amino-6-(2,4-dimethoxyphenyl)-4-(1,5-dimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-N-(2,2,2-trifluoroethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(2-ethylphenyl)-6-methylpyridin-2-amine
5-(2-chloro-4-fluorophenoxymethyl)-N-[2-(pyridin-3-yl)ethyl]-1,2-oxazole-3-carboxamide
3-[(2-cyclohexylpyrimidin-5-yl)methyl]-9-methyl-3,9-diazaspiro[5.6]dodecan-10-one
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamide
3-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylpyridazine
N-cyclopropyl-1-{1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
N-methyl-4-[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1,3-thiazol-2-amine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
1-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
9-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
ethyl 1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
8-methoxy-2-{[4-(4-methoxyphenyl)piperazin-1-yl]methyl}quinoline
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
5-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]quinoxaline
4-(4-methylpiperazin-1-yl)-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}benzamide
3-{1-[4-(4-chlorophenyl)butanoyl]piperidin-4-yl}-1,3-oxazolidin-2-one
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-(4-propanoylphenoxy)acetamide
2-[2-methyl-3-(4-phenyl-1H-imidazol-5-yl)-1H-indol-1-yl]acetamide
1-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}cyclopropane-1-carboxamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(6-methylpyridine-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-cyclobutyl-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
2-(3-methoxypropyl)-9-(2-phenylacetyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(5-ethyl-1,2,4-oxadiazol-3-yl)-4-[(4-fluorophenyl)methyl]-1,4-diazepane
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-{[(4-methylphenyl)amino]methyl}benzamide
(2R,3S,6R)-5-(2-ethylpyridine-4-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
(2S,4S)-4-amino-N-(1-ethynylcyclohexyl)-1-methylpyrrolidine-2-carboxamide
[(3R,4R)-1-(3,4-difluorobenzoyl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
5-(1,3-benzothiazole-6-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
(2R,3S,6R)-5-(2-ethoxypyridine-3-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N,3-dimethyl-N-[(3-methylthiophen-2-yl)methyl]-1-propyl-1H-pyrazole-4-carboxamide
2-chloro-N-[1-(methylcarbamoyl)cyclohexyl]-5-(1H-pyrazol-1-yl)benzamide
6-[(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-2-oxo-decahydro-1,6-naphthyridin-6-yl]pyridine-3-carbonitrile
7-[(3-benzyl-1H-1,2,4-triazol-5-yl)methoxy]-4-ethyl-2H-chromen-2-one
1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethan-1-one
1-(2,5-dimethylfuran-3-carbonyl)-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine