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5-ethanesulfonamido-N,1-dimethyl-2-phenyl-N-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
6-methyl-2-{[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]amino}pyridine-3-carbonitrile
2-hydroxy-N-methyl-3-(2-methylphenoxy)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
5-{4-[2-fluoro-6-(propan-2-yloxy)phenyl]phenyl}-1H-1,2,3,4-tetrazole
1-(3,5-dichloro-4-methylbenzoyl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
2-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-[(1-methylpiperidin-3-yl)methyl]-1,3-oxazole-4-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
N-({7-[2-(1H-pyrazol-1-yl)butanoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
8-[(1-methyl-1H-indol-3-yl)methyl]-1-(3-methylbutyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetyl]-4-(4-methylphenoxy)piperidine-4-carboxylic acid
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carboxamide
(4aS,7aR)-1-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-methoxy-3-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)-1-benzofuran-2-carboxamide
1-{1-[4-(4-methylphenyl)phenyl]piperidin-4-yl}piperidin-4-ol
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
2-(4-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}piperazin-1-yl)pyrazine
methyl 1-(2-methylpropyl)-3-(2-phenylacetamido)-5-{[1-(pyridin-3-yl)propan-2-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(1R,5R)-3-(3-fluoro-4-methylbenzenesulfonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
5-(3-benzyl-1H-1,2,4-triazol-5-yl)-1-propylpiperidin-2-one
1-[3-({[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenyl]ethan-1-one
4-(3-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}propoxy)benzamide
(2R)-2-acetamido-N-[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]butanamide
N-[(1,4-dimethylpiperazin-2-yl)methyl]-5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-methyl-N-[(4-methylphenyl)methyl]acetamide
(3S,4R)-4-phenyl-1-{2-[(thiophen-2-ylmethyl)carbamoyl]ethyl}pyrrolidine-3-carboxylic acid
2-(naphthalen-2-yloxy)-1-[4-(pyridin-3-yl)piperazin-1-yl]propan-1-one
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-1-(oxan-4-yl)piperidine-4-carboxamide
N-(dicyclopropylmethyl)-N-methyl-9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
1,3-dimethyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-pyrazole-4-carboxamide
(1S,5R)-3-(1-benzofuran-2-ylmethyl)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2,7,8-trimethyl-4-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]quinoline
1-(1-ethyl-1H-1,2,3-triazol-4-yl)-3-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]urea
N-{1-[(2-fluorophenyl)methyl]-1H-pyrazol-4-yl}-3-[(methylsulfanyl)methyl]piperidine-1-carboxamide
2-(morpholin-4-yl)-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]pyrimidine-5-carboxamide
2-(methylsulfanyl)-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
2-{3-cyclopentyl-5-[2-(1H-indol-3-yl)ethyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
1-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
4-(cyclopropylmethyl)-1-(3-phenyl-1,2-oxazole-4-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-methyl-N-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide
[1-(1-benzothiophen-2-ylmethyl)-4-benzylpiperidin-4-yl]methanol
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-phenylpiperidin-4-ol
2-(3-acetyl-1H-indol-1-yl)-N-cyclopropyl-N-(pyridin-2-ylmethyl)butanamide
4-[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]piperidine
1-{[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(3-methylphenoxy)piperidine
(3S,5S)-1-methyl-5-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrrolidin-3-amine
[(3R,4R)-1-(6-cyclopropylpyrimidin-4-yl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
2-(2-chloro-6-fluorophenyl)-1-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}ethan-1-one
5-butyl-1-(2-methoxyphenyl)-4-(4-methylpyrimidine-5-carbonyl)piperazin-2-one