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2,2-diethyl-4-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}morpholine
N-[(3,4-difluorophenyl)methyl]-3-[1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-3-yl]propanamide
(1R,5S,6R)-3-(1,3-dihydroxypropan-2-yl)-N-(9H-fluoren-9-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide
3-amino-1-{[3-methoxy-4-(pyrrolidin-1-yl)phenyl]methyl}pyrrolidine-3-carboxylic acid
2-(dimethylamino)-7-(oxane-2-carbonyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]-4-(1H-pyrrole-2-carbonyl)piperazine
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
6-{[(1R,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]cyclohex-3-ene-1-carboxamide
3-(5-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
2-(2,4-dimethylphenyl)-2-{methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}acetic acid
1-{[2-(3-hydroxypiperidin-1-yl)-6-methylquinolin-3-yl]methyl}-1,4-diazepan-5-one
2-methyl-5-{4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
N2-[2-(dimethylamino)-1-phenylethyl]-N4,N4,5-trimethylpyrimidine-2,4-diamine
1-[1-(4-fluorophenyl)-2,2-dimethylcyclopropanecarbonyl]-4-(thian-4-yl)piperazine
1-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
4-methyl-2-{[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]methyl}-5,6,7,8-tetrahydroquinazoline
(3S,4S)-3-hydroxy-N-(1-methyl-3-phenyl-1H-pyrazol-5-yl)-4-(morpholin-4-yl)pyrrolidine-1-carboxamide
6-[7-(oxan-4-yl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]pyridine-3-carbonitrile
1-(2,3-dihydro-1H-inden-2-yl)-N-[2,2-dimethyl-3-(morpholin-4-yl)propyl]-N-methylpiperidin-3-amine
5-methoxy-N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)-1H-indole-2-carboxamide
1-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)-4-(piperidine-1-carbonyl)piperidine
5-{[2-(4-methylpentyl)morpholin-4-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(1S,4S)-5-benzyl-2,5-diazabicyclo[2.2.1]heptan-2-yl]-2-(7-fluoro-2-methyl-1H-indol-3-yl)ethan-1-one
{1-[6-amino-2-(morpholin-4-yl)pyrimidin-4-yl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
N-(1-{1-[2-(2-chlorophenoxy)acetyl]piperidin-4-yl}-2-(4-fluorophenyl)ethyl)-2-(dimethylamino)-N-methylacetamide
4-hydroxy-1-(5-propyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)piperidine-4-carboxylic acid
4-(3-chloropyridin-2-yl)-1-[(4-methoxyphenyl)methyl]piperazin-2-one
2-(4-fluorophenyl)-1-[2-(1H-pyrazol-1-yl)benzoyl]piperidine
2-(2,5-dioxoimidazolidin-1-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)acetamide
4-[1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]thiomorpholine
2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepine
methyl 6-[1-(cyclohexylmethyl)-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl]pyridine-2-carboxylate
5-fluoro-3-methyl-N-[2-(1-methylpiperidin-3-yl)ethyl]-1H-indole-2-carboxamide
6-(3-hydroxypiperidin-1-yl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
2-(3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}pyrrolidin-1-yl)-5-(trifluoromethyl)pyridine
3-[(4-fluorophenyl)formamido]-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]propanamide
1-(5-ethyl-1,2-oxazole-4-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
3-(ethoxymethyl)-1-(2-methoxyphenyl)-5-methyl-1H-1,2,4-triazole
2-(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidin-3-yl)benzoic acid
N-(2-methylpropyl)-N-[(3-methylthiophen-2-yl)methyl]pent-4-ynamide
2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)benzamide
1-methyl-8-[1-(methylsulfanyl)propan-2-yl]-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(dimethyl-1,2-oxazol-4-yl)-3-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1H-pyrrole-2-carboxamide
2-[(2-chlorophenyl)methyl]-4-(thiophene-3-carbonyl)morpholine
(2E)-N-({3-methyl-7-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-(thiophen-2-yl)prop-2-enamide
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
3-(5-cyclohexyl-1,3,4-oxadiazol-2-yl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
14-ethyl-5-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one