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(2S,4R)-4-(cycloheptylamino)-N-ethyl-1-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxamide
N-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
1,3-dimethyl-6-(pyridin-2-yl)-N-[1-(pyridin-4-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(2S,4R,6S)-2-(1,5-dimethyl-1H-pyrazol-4-yl)-6-(2-phenylethyl)oxan-4-yl]acetamide
N-{[1-(ethanesulfonyl)piperidin-3-yl]methyl}-3,5-dimethoxybenzamide
3-{6-oxa-9-azaspiro[4.5]decan-9-ylmethyl}pyridin-2-amine
2-{1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,3-triazol-4-yl}-8-methoxyquinoline
ethyl 4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
8-[(3-hydroxyphenyl)methyl]-1-methyl-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(2-amino-5-ethylpyrimidin-4-yl)amino]-N-methylpentanamide
1-ethyl-3-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyrrolidine
7-(5-chloropyridin-2-yl)-4-(2-hydroxybutyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(2-methoxy-4-{[methyl(pyrimidin-4-ylmethyl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
5-cyclopropyl-N-(2-methoxyethyl)-1-[4-(3-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
2-methyl-6-(3-{[4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)-2,3-dihydropyridazin-3-one
4-[(2-methylpyridin-3-yl)oxy]-1-(4-methylpyrimidin-2-yl)piperidine-4-carboxylic acid
3-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-4,5,6,7-tetrahydro-1-benzofuran-4-one
(1S,5R)-6-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-{5-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidine-1-carbonyl]-2-methylphenyl}imidazolidin-2-one
3-{2-[4-(4-methylphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-1λ6-thiolane-1,1-dione
dimethyl(3-{2-[1-(6-methylpyridazin-3-yl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
7-(2,6-difluoro-3-methylbenzoyl)-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
5-cyclopropanecarbonyl-1'-[(2-fluoro-5-methylphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{2-[1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-2-yl]ethyl}pyridine
1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-methylbut-2-en-1-one
N-(2,3-dihydro-1H-inden-2-yl)-N-propyl-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
1-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}cyclopropane-1-carboxamide
1-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
2-(morpholin-4-yl)-2-(pyridin-3-yl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}acetamide
2-ethyl-5-[3-(3-methoxypropyl)piperidine-1-carbonyl]pyrimidine
(1S,6R)-9-[(2,3-dimethyl-1H-indol-7-yl)methyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
2-{[(1-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
diethyl({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)amine
N-[2-(benzylsulfanyl)ethyl]-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-2-methoxyethan-1-one
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[2-(1H-indol-3-yl)ethyl]-1,3-oxazole-4-carboxamide
6-{2-[2-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
(1S,5R)-6-(5-methylpyrazine-2-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
5-[(dimethylamino)methyl]-N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]-1,3,4-oxadiazole-2-carboxamide
N-(3-chloro-4-methoxyphenyl)-3-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-yl)propanamide
4-{4-[4-(2-methoxyethoxy)phenyl]phenyl}morpholine
4-benzyl-1-(3,5-difluoropyridine-2-carbonyl)-3-ethyl-1,4-diazepan-5-one
(3S)-1-benzyl-N-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]pyrrolidin-3-amine
2-(2-cyclopropylpyrimidin-5-yl)-6-fluoro-4-(morpholine-4-carbonyl)quinoline
2-{4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-5-methylpyrazine
(4S)-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
N-(5-methanesulfonamido-2-methylphenyl)-2-(methoxymethyl)piperidine-1-carboxamide
methyl 3-[(3S,4R)-1-[(2-methoxynaphthalen-1-yl)methyl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]propanoate
(1S,5R)-6-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(2-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-2-yl}ethyl)pyridine