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5-(4-chloro-2-methoxyphenoxymethyl)-N-[(2S)-1-hydroxypropan-2-yl]-1,2-oxazole-3-carboxamide
2-cyclopropyl-1-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}ethan-1-one
2-(2-fluorophenoxymethyl)-N-[(3-methoxyphenyl)methyl]-1,3-oxazole-4-carboxamide
2-[1-(2-methylpropyl)-4-[(2,4,6-trimethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
1-{4-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]piperidin-1-yl}ethan-1-one
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}dimethylamine
1-{6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carbonyl}piperidine
2-(dimethyl-1,3-thiazol-5-yl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)propanamide
1-(3-fluorobenzoyl)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(2S)-2-[3-(1,2-oxazinan-2-yl)propanamido]-3-phenylpropanoic acid
(3aS,6aS)-2-[1-(3-chloro-4-methylphenyl)piperidin-4-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(4aR,8aR)-4a-hydroxy-7-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
(2S)-4-methyl-2-({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amino)pentanamide
1-{2-[3-cyclopropyl-1-(4-methoxyphenyl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,3,4-tetrazole
4-(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}pyrrolidin-3-yl)-2-(pyridin-4-yl)pyridine
2-ethoxy-5-(2-{methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}pyrimidin-4-yl)benzoic acid
4-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1-oxaspiro[4.4]nonan-2-one
1-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-4-[3-(4-fluorophenoxy)propyl]piperazine
4-{4-[(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)amino]piperidin-1-yl}-6-methylpyrimidin-2-amine
1-[1-(2-fluorophenyl)cyclopropaneamido]cyclopentane-1-carboxamide
5-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-N,N-dimethylpyridin-2-amine
1-(3-methylcinnolin-5-yl)-3-{2-[(trifluoromethyl)sulfanyl]ethyl}urea
4-(5-{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
1-(2-cyanobenzoyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-[3-(3-methyl-1H-pyrazol-1-yl)propyl]-6-(propan-2-yl)pyrimidin-4-amine
3-{3-[1-(dimethylamino)ethyl]phenyl}-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
3-({1-ethyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}methyl)adamantan-1-ol
2-[4-(3-methoxyphenyl)-3-oxopiperazine-1-carbonyl]benzonitrile
2-(1-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1H-imidazol-2-yl)-4,5,6,7-tetrahydro-1,3-benzothiazole
N-{[5-({[(4-fluorophenyl)methyl](prop-2-en-1-yl)amino}methyl)furan-2-yl]methyl}-N-methylmethanesulfonamide
2-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]acetic acid
5-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-(dimethylamino)butanamide
2-(2-methoxyethyl)-9-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-2,9-diazaspiro[5.5]undecan-3-one
4-[1-benzyl-5-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
8-chloro-2-methyl-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}quinoline-4-carboxamide
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)[2-methyl-2-(morpholin-4-yl)propyl]amine
5-methanesulfonyl-2-methyl-N-[(1-methyl-1H-imidazol-2-yl)(phenyl)methyl]pyrimidin-4-amine
3-(1H-pyrazol-1-ylmethyl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}benzamide
N,6-dimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-oxo-2-(2-phenylethyl)-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
1-[9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(3,4,5-trimethoxyphenyl)ethan-1-one
(3S,4S)-4-cyclopropyl-1-[2-(methylamino)-1,3-thiazole-4-carbonyl]pyrrolidine-3-carboxylic acid
1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
methyl 3-[(3S,4R)-1-{[3-(benzyloxy)phenyl]methyl}-4-(morpholin-4-yl)piperidin-3-yl]propanoate
1-benzyl-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
5-(2-chloro-4-fluorophenoxymethyl)-3-(1,2-oxazolidine-2-carbonyl)-1,2-oxazole
2-ethyl-8-[3-(methylsulfanyl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
4-(2-hydroxy-4-methylpentanoyl)-1-phenylpiperazin-2-one
4-methoxy-2-{[9-methoxy-7-(8-methoxy-4-methylquinolin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenol