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2-(4-fluorophenyl)-1-(3-methoxypropyl)piperidine
2-amino-4-methyl-N-[2-(pyridin-3-yloxy)propyl]-1,3-thiazole-5-carboxamide
1-(5-ethyl-2-methylpyrimidin-4-yl)-N-methylpyrrolidine-3-carboxamide
8-(ethanesulfonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
6-[9-oxo-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-3-carbonitrile
5-[1-(1,2-oxazole-3-carbonyl)pyrrolidin-2-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]thiophene-2-carboxamide
2-(3-methyl-1H-pyrazol-1-yl)-1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-[(2-ethoxyphenyl)methyl]-N-ethyl-2-(4-ethylpiperazin-1-yl)acetamide
3-(5-cyclobutyl-1,3,4-thiadiazol-2-yl)-1-{[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}urea
6-(azepane-1-carbonyl)-N-(2H-1,3-benzodioxol-5-ylmethyl)-5-methylthieno[2,3-d]pyrimidin-4-amine
2,4-dimethyl-6-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyrimidine
N-(2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)methanesulfonamide
N-cyclopropyl-2-{6-[(pyridin-4-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
3-(4-chloro-1H-pyrazol-1-yl)-1-[3-(2-methoxyphenoxy)azetidin-1-yl]propan-1-one
3-[3-(2-methylphenoxy)azetidine-1-carbonyl]-2-(methylsulfanyl)pyridine
butyl 9-oxo-8-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecane-2-carboxylate
1-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
1-[4-(morpholine-4-carbonyl)phenyl]-N-(propan-2-yl)piperidin-4-amine
3-(furan-2-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
7-{[2-(propylsulfanyl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decane
(3aS,6aR)-2-oxo-N-(propan-2-yl)-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carboxamide
2-(5-{1-[cyclohexyl(methyl)amino]ethyl}-1H-1,2,4-triazol-1-yl)ethan-1-ol
7-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-amino-4-(3,4-dihydroxyphenyl)-6-(2,2-dimethylcyclopropyl)-5-methylpyridine-3-carbonitrile
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)(pyridin-3-ylmethyl)amine
N-[(2-chlorophenyl)methyl]-3-[1-(1H-1,2,4-triazole-5-carbonyl)piperidin-3-yl]propanamide
2-({2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}methyl)pyridine-3-carboxylic acid
1-(isoquinoline-1-carbonyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
2-[(5-{[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]methyl}pyrimidin-2-yl)(methyl)amino]acetic acid
5-{3-oxo-3-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]propyl}imidazolidine-2,4-dione
2-amino-N-({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
7-(3-chlorophenyl)-4-(pyridine-3-carbonyl)-9-(thiophen-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[5-(2-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
3-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidine-1-carbonyl]-1-methyl-6-(propan-2-yl)-1,2-dihydropyridin-2-one
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N,2,2-trimethyl-1-(thiophen-2-yl)cyclopropane-1-carboxamide
N,7,8-trimethyl-2-(1-methyl-1H-pyrazol-4-yl)-N-[1-(pyridin-4-yl)ethyl]quinoline-4-carboxamide
5-{[(propan-2-yl)({[3-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}pyrrolidin-2-one
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-(1-phenylcyclopropyl)benzamide
N-{[3-methyl-7-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
1-(2-{3-benzyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}ethyl)-4-chloro-1H-pyrazole
1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-[(3-methylphenyl)sulfanyl]piperidine
4-[({5-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}sulfanyl)methyl]pyridine
1'-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(2,5-difluorophenyl)methyl]-3-(1,3-dimethyl-1H-pyrazol-5-yl)-1-(1-methoxypropan-2-yl)urea
(3S,4S)-4-cyclopropyl-1-[4-(morpholin-4-yl)benzoyl]pyrrolidine-3-carboxylic acid
N-(4-methoxyphenyl)-2-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]butanamide
2-[(3,5-difluorophenyl)methyl]-8-(oxolane-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1'-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
4-(4-fluoro-2-methylphenoxy)-1-(furan-2-carbonyl)piperidine-4-carboxylic acid
N-{2-[2-(adamantan-1-yl)-6-oxo-1,6-dihydropyrimidin-4-yl]ethyl}acetamide