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{3-[(2-methylphenyl)methyl]-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-3-yl}methanol
(3S,4S)-1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperidine-3,4-diol
2-ethyl-5-{[4-(2-methoxyphenoxy)piperidin-1-yl]methyl}pyrimidine
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-phenylprop-2-ynamide
1-[2-(dimethylamino)-4-{[3-(2-methyl-1H-imidazol-1-yl)propyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1-ethyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-1H-pyrazole-4-sulfonamide
1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-4-(3-methylphenoxy)piperidine-4-carboxylic acid
1-(2-fluorophenyl)-4-[(3-{[1-(3-methylthiophene-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(6-methylpyridazin-3-yl)pyrrolidin-3-yl]methanol
3-({2-[1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}(methyl)amino)-1λ6-thiolane-1,1-dione
2-(1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1H-pyrazol-4-yl)ethan-1-ol
6-(2-methylpyrrolidin-1-yl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1,4-dioxane-2-carboxamide
3-{[methyl({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amino]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-hydroxy-3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
1-[2-(4-chlorophenyl)morpholin-4-yl]-2-(3-hydroxyphenyl)ethan-1-one
(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-1-[(3,4-dimethoxyphenyl)methyl]-N-[(2-methoxyphenyl)methyl]piperidine-3-carboxamide
5-[(5-methylthiophen-2-yl)sulfonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
(4aS,8aS)-2-cyclopentanecarbonyl-7-(2-methylpyrimidine-5-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
4-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}pyrimidin-2-amine
3-(1-butyl-1H-imidazol-2-yl)-1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine
N-(3-hydroxypropyl)-N-methyl-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
3-(2,6-dimethoxyphenyl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
6-{6-[3-(dimethylamino)propoxy]pyridin-3-yl}pyridin-3-amine
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-5-(1H-indol-1-ylmethyl)-N-methyl-1H-pyrazole-3-carboxamide
1-(3-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}piperidin-1-yl)propan-1-one
2-{[1-(2-ethylpyrimidine-5-carbonyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
N-{[5-(2-chlorophenyl)-1,2-oxazol-3-yl]methyl}-5-cyclobutyl-1,3,4-oxadiazol-2-amine
5-(methoxymethyl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]furan-2-carboxamide
4-[(4aR,7aS)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N-cyclopentyl-4-oxobutanamide
2-[(2-{9-hydroxy-1,5,7-trimethyl-3,7-diazabicyclo[3.3.1]nonane-3-carbonyl}phenyl)amino]acetic acid
1-methyl-4-oxo-N-(pentan-3-yl)-N-(2-phenylethyl)-1,4-dihydroquinoline-3-carboxamide
N-[3-(3-methylphenyl)phenyl]-1-(pyrazine-2-carbonyl)pyrrolidine-2-carboxamide
2-cyclopentyl-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)acetamide
7-[(2,3-difluorophenyl)methyl]-2-(4-methyl-1H-imidazole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-[1-(furan-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-2-methylphenol
1-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2-methyl-4-phenylpiperazine
1-{2-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
5-fluoro-N4,N4-dimethyl-N2-[2-(4-phenylpyrimidin-2-yl)ethyl]pyrimidine-2,4-diamine
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-4-(piperidin-3-yl)benzamide
N-phenyl-1-{2-[(2,3,4-trimethoxyphenyl)formamido]ethyl}-1H-1,2,3-triazole-4-carboxamide
(2S,4R)-1-(4-chloro-1H-pyrazole-3-carbonyl)-N,N-diethyl-4-propanamidopyrrolidine-2-carboxamide
2-(1-{[1-(1-benzylpyrrolidin-3-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-amine
methyl 2-[3-(2-ethylphenoxy)azetidine-1-carbonyl]piperidine-1-carboxylate
3-{1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{3-[(2,4-difluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}-2-methoxyethan-1-one
1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
3-methyl-N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
4-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-cyclohexyl-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one