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6-{2-[bis(propan-2-yl)carbamoyl]phenyl}pyridine-2-carboxamide
9-[3-(2-methoxyphenyl)propanoyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
6-(benzyloxy)-1-(2-methylpropyl)-4-(thiophene-3-carbonyl)-1,4-diazepan-2-one
1-(5-phenyl-1,2,4-oxadiazol-3-yl)-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
N-{1-[1-(2-methoxybenzoyl)piperidin-4-yl]-2-phenylethyl}-N-methylthiophene-3-carboxamide
6-{3-oxo-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-3-carbonitrile
2-(3-{3-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]phenyl}-1H-pyrazol-1-yl)ethan-1-ol
N-ethyl-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
3-(2H-1,3-benzodioxol-5-yl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}propanamide
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-({[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}amino)pyridine-3-carboxamide
1-(2-{1-[5-(methoxymethyl)thiophene-2-carbonyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
1-cycloheptyl-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
N-(3-methylphenyl)-3-[1-(quinoline-8-sulfonyl)piperidin-4-yl]propanamide
1-(5-ethyl-1,3-oxazole-4-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
N-(2,5-difluorophenyl)-5-oxo-1,4,9-triazaspiro[5.5]undecane-9-carboxamide
2-[(2E)-3-phenylprop-2-en-1-yl]-8-[(2R)-pyrrolidine-2-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-(morpholin-4-yl)pyrimidine-5-carboxamide
(1S,5R)-3-[4-(4-methoxyphenyl)butanoyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{[(1-cyclopentanecarbonylpiperidin-4-yl)formamido]methyl}benzoic acid
2-(2,3-dihydro-1H-inden-1-yl)-N-[3-(4-methylpiperazin-1-yl)propyl]acetamide
1-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-methyl-3-(1H-pyrazol-1-yl)propan-1-one
N-(2-methoxyethyl)-6-[4-(2-methoxyethyl)piperazine-1-carbonyl]-5-methylthieno[2,3-d]pyrimidin-4-amine
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]benzamide
3-hexyl-8-(2-methylpyrimidine-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-methyl-4-{5-[1-(4-methylphenyl)-1H-pyrazol-4-yl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}piperidine
1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4-(pyridin-2-ylmethyl)-1,4-diazepane
5-(3-cyclohexyl-1H-pyrazol-4-yl)-4-phenyl-1-(pyrrolidin-3-yl)-1H-imidazole
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}benzamide
5-[1-(5-methoxy-1-methyl-1H-indole-2-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
(9aS)-2-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine
N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
2-(hydroxymethyl)-N-(3-phenylphenyl)piperidine-1-carboxamide
N-(1-hydroxybutan-2-yl)-2-oxo-N-(pyridin-2-ylmethyl)pentanamide
5-butyl-1'-(2,5-dimethylfuran-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}acetamide
4-{[7-(2-hydroxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]methyl}-1-methyl-1H-pyrrole-2-carbonitrile
(2R,6R)-4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
5-(2,4-difluorophenoxymethyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-{[5-(4-cyanophenyl)-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
7-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[(prop-2-en-1-yl)amino]methyl}piperidin-2-one
methyl 3-[(3S,4R)-1-[(3-ethoxy-2-hydroxyphenyl)methyl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]propanoate
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)(3-phenylpropyl)amine
2-amino-4-(3-chloro-4-hydroxy-5-methoxyphenyl)-6-(3,5-dimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
2-{5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-yl}benzoic acid
1-ethyl-N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-[(2-chlorophenyl)methyl]-4-{4-[(4-fluorophenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-[1-(thian-4-yl)piperidin-4-yl]propanamide