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(4aS,8aS)-2-[4-(propan-2-yl)pyrimidin-2-yl]-decahydro-2,7-naphthyridin-4a-ol
3-methoxy-5-(2-methylpyrrolidine-1-carbonyl)benzoic acid
4-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-1-phenylpiperazin-2-one
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-2-(methylamino)pyridine-4-carboxamide
2-ethyl-5-[1-ethyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]pyrimidine
5-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)-2,2-dimethylpentan-1-ol
(1R,9S)-5-amino-3-(4-hydroxynaphthalen-1-yl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N,1,3-trimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(2S,4S)-4-amino-1-[(4-methanesulfonylphenyl)methyl]-N-methylpyrrolidine-2-carboxamide
1-methyl-3-(propan-2-yl)-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}-1H-pyrazole-5-carboxamide
(1S,5R)-6-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
1-{[6-(2,6-dimethoxyphenyl)pyridin-3-yl]methyl}-4-methylpiperazine
N-methyl-4-{[(3-methylthiophen-2-yl)methyl]amino}-N-(prop-2-yn-1-yl)benzamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-2-(1H-pyrazol-1-yl)butanamide
[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]({[3-(1H-pyrazol-1-yl)phenyl]methyl})amine
4-(5-fluoro-2-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}pyrimidin-4-yl)morpholine
2-(5-{2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]ethyl}-3-(3-fluorophenoxymethyl)-1H-1,2,4-triazol-1-yl)ethan-1-ol
2-acetamido-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
5-{3-cyclopentyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1-methyl-3-propyl-1H-pyrazole
6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-2-ol
N-(1-hydroxybutan-2-yl)-2-(1-propylpiperidin-4-yl)-N-(pyridin-2-ylmethyl)acetamide
1-[3-(methylsulfanyl)butyl]-4-(1H-pyrazol-3-yl)piperidine
5-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenoxy]-1-azabicyclo[3.2.1]octane
1-[1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
1-(3-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(methylamino)ethan-1-one
1-cyclopentanecarbonyl-N-[(5-fluoro-2-methylphenyl)methyl]piperidine-4-carboxamide
3,5-dimethyl-4-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-2-yl)-1,2-oxazole
N-{1-[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
2-[(1S,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetic acid
2-ethoxy-5-(2-{[(1-methylpyrrolidin-3-yl)methyl]amino}pyrimidin-4-yl)benzoic acid
N-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidine-1-carboxamide
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(methoxymethyl)-1H-1,2,4-triazole
N-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}-2-(morpholin-3-yl)acetamide
3-{1-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-1-oxopropan-2-yl}-3,4-dihydroquinazolin-4-one
6-methyl-5-{5-[2-(pyrrolidin-1-yl)phenyl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(4-methoxyphenoxy)piperidine
3-methyl-8-{[5-(oxan-2-yl)furan-2-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-(2-methoxyethyl)-2-[(1-methyl-1H-pyrazol-4-yl)methyl]-2,7-diazaspiro[4.5]decane
{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
4-[(5-{1-[(4-methoxypyridin-2-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]morpholine
3-[(4-propylpiperazin-1-yl)methyl]-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
N-{1-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
3-(3-methyl-3-phenylpiperidin-1-yl)propanamide
(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)[(3-methyl-1H-indol-2-yl)methyl]amine
1-({1-[(4-fluorophenyl)methyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}methyl)-1,2-dihydropyridin-2-one
5-butyl-1-(4-chlorophenyl)-4-(1H-pyrrole-2-carbonyl)piperazin-2-one
1-{1'-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
3-{[(dicyclopropylmethyl)amino]methyl}-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
methyl 6-[(2,4-difluorophenyl)methyl]-2-(phenylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(4-chlorophenyl)-N-{[4-(4-fluorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}cyclopropane-1-carboxamide