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8-fluoro-2-({4-[(methylsulfanyl)methyl]piperidin-1-yl}methyl)quinolin-4-ol
(4aS,8aR)-1-(2-aminoethyl)-6-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-decahydro-1,6-naphthyridin-2-one
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl){[3-(morpholin-4-ylmethyl)phenyl]methyl}amine
1-(oxane-4-carbonyl)-3-(2-phenylethyl)piperidine
[(5-methylthiophen-2-yl)methyl](prop-2-en-1-yl)(pyridin-3-ylmethyl)amine
methyl({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)[(3-methylthiophen-2-yl)methyl]amine
2-(3-{[3-(piperidin-1-ylmethyl)piperidin-1-yl]methyl}phenyl)ethan-1-amine
3-(3-hydroxyquinoxalin-2-yl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]propanamide
N-(1-benzylpiperidin-4-yl)-5-(propan-2-yl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-2-(methylsulfanyl)benzamide
1-cyclopentyl-N-ethyl-5-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
3-(2,5-dimethoxyphenyl)-1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)pyrrolidine
N'-[1-(4-chlorophenyl)-3-hydroxypropan-2-yl]-N-(2,4-dimethoxyphenyl)propanediamide
1-ethyl-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
2-cyclopentyl-9-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2,9-diazaspiro[5.5]undecan-3-one
5-[4-(2-chlorophenoxy)piperidine-1-carbonyl]-2-cyclopropyl-3,4-dihydropyrimidin-4-one
5-ethyl-6-methyl-N4-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}pyrimidine-2,4-diamine
3-{[1-(2-methoxypyridine-3-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
2-[4-(4-ethylpiperazine-1-carbonyl)-5-(furan-2-yl)-1H-pyrazol-1-yl]-4-(2-methoxyphenyl)pyrimidine
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-1-phenylcyclopropane-1-carboxamide
5-methyl-5-(4-methylpent-3-en-1-yl)-1-[(5-methylpyrazin-2-yl)methyl]piperidin-2-one
5-(3,5-dimethylfuran-2-carbonyl)-3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-ethoxy-5-[2-(2-methylbutyl)pyrimidin-4-yl]benzoic acid
3-[2-oxo-2-(3-oxo-4-phenylpiperazin-1-yl)ethyl]imidazolidine-2,4-dione
4-[4-(benzenesulfonyl)piperazin-1-yl]-2-methoxypyridine-3-carbonitrile
N-methyl-6-(piperidin-4-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)pyrimidin-4-amine
N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-2-(pyridin-4-ylsulfanyl)acetamide
4-benzyl-2-{2-[7-(5-chloro-2-methoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
N-[(5,6-dimethylpyridin-3-yl)methyl]-4-(3-hydroxy-3-methylbutyl)benzamide
3-{[(3R,4S)-3-(2-carboxyethyl)-4-(dimethylamino)piperidin-1-yl]sulfonyl}thiophene-2-carboxylic acid
1-(2-chlorophenyl)-3-{1-[1-(5-methylhex-5-en-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
ethyl 2-[4-(3-methylpyridin-2-yl)piperazin-1-yl]acetate
N-[(3R,4S)-1-(4-chloro-3-fluorobenzoyl)-4-propylpyrrolidin-3-yl]acetamide
methyl 4-(5-{[benzyl(2-hydroxyethyl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
N-[1-(5-{[2-(4-fluorophenoxy)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(3-fluorophenyl)benzamide
(2S,4R)-4-amino-1-{[1-(4-cyanophenyl)-1H-pyrrol-2-yl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-[2-methoxy-4-({[(5-methylfuran-2-yl)methyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
3-(1-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}piperidin-2-yl)propan-1-ol
N-[2-(diethylamino)ethyl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-3-[4-(3-methylphenyl)piperazin-1-yl]propan-1-one
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
3-(3-methoxyphenoxymethyl)-1-(3-methyl-1H-pyrazole-5-carbonyl)piperidine
1-(pyridin-4-ylmethyl)-4-[4-(1H-1,2,4-triazol-1-yl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-[(4-{4-[(4-chlorophenyl)methyl]piperazine-1-carbonyl}phenyl)sulfanyl]ethan-1-ol
2-hydroxy-3-(2-methylphenoxy)-1-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propan-1-one
N,N-dimethyl-3-[(2-oxo-1,2,3,4-tetrahydroquinolin-1-yl)methyl]-1,2,4-oxadiazole-5-carboxamide