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3-(propan-2-yl)-4-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperazin-2-one
3-{1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
5-methyl-3-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-butyl-8-(2-fluoro-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{6-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]-2-methylpyrimidin-4-yl}ethan-1-amine
1-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-ethoxyethan-1-one
6-(azocane-1-carbonyl)-N-(furan-2-ylmethyl)-5-methylthieno[2,3-d]pyrimidin-4-amine
N-ethyl-1-[3-(3-hydroxy-3-methylbutyl)benzoyl]pyrrolidine-3-carboxamide
4-(4-fluorophenyl)-1-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}-1,2,3,6-tetrahydropyridine
2-{1-[(4-ethoxyphenyl)methyl]-4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperazin-2-yl}ethan-1-ol
methyl[(3-methylthiophen-2-yl)methyl][1-(pyridin-2-yl)ethyl]amine
3-(1-cyclopentyl-1H-pyrazol-5-yl)-1-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)urea
1-[(3,4-difluorophenyl)methyl]-3-(2-methoxyphenoxy)azetidine
6-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
2-methyl-4-{3-[4-(pyrrolidin-1-yl)piperidine-1-carbonyl]phenyl}butan-2-ol
3-{2,7-diazaspiro[4.5]decane-2-carbonyl}-2-methyl-N-(pyridin-2-ylmethyl)aniline
N-ethyl-N-methyl-2-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}acetamide
4-(trifluoromethyl)-1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-(2-methoxyphenyl)-N-methyl-1H-pyrazole-4-carboxamide
[(3S,5R)-5-[(dimethylamino)methyl]-1-(5-methyl-2-phenylfuran-3-carbonyl)piperidin-3-yl]methanol
4-[(3S,4R)-4-amino-3-methoxypiperidin-1-yl]-6-methylpyrimidin-2-amine
1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-[4-(1H-imidazol-1-yl)phenyl]-1H-imidazole
N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-N-(oxolan-3-ylmethyl)cyclopentanamine
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-{2-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl}piperazine
N-[2-(dimethylamino)ethyl]-N-methyl-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
[(2,4-difluoro-3-methoxyphenyl)methyl](methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
N-{1-[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
N-(3-hydroxy-3-phenylpropyl)-N-methyl-2-(methylamino)pyrimidine-5-carboxamide
N-[2-(3-methoxypropanoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-4-(trifluoromethyl)benzamide
N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
1-[(5-chloro-3-methyl-1H-indol-2-yl)methyl]-3-(hydroxymethyl)piperidin-3-ol
3-(3-methanesulfonamido-4-methoxyphenyl)-1-[1-(pyrazin-2-yl)propan-2-yl]urea
1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
2-(2H-1,2,3-benzotriazol-2-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-[(E)-2-phenylethenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-[(2-methyl-1,3-thiazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
2-chloro-4-({[1-(oxan-4-yl)piperidin-4-yl]carbamoyl}amino)benzamide
3-[(2R,3R,6R)-5-[1-(methoxymethyl)cyclobutanecarbonyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
(3aS,6aS)-1-(3-chloro-4-fluoro-1-benzothiophene-2-carbonyl)-octahydropyrrolo[2,3-c]pyrrole
5-{1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]pyrrolidin-2-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-5-propyl-1,2-oxazole-4-carboxamide
2-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-1,3-dimethyl-1H-indole
ethyl({[(1R,5S,6R)-3-(2-methylbenzoyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl})(oxan-4-ylmethyl)amine
2-(6-methoxypyridin-3-yl)-2-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}acetic acid
2-[2-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl]pyridin-3-ol
2-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-N-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
{[2-(3-chlorophenyl)-6,7-dimethoxyquinolin-3-yl]methyl}(2-methoxyethyl)methylamine
1-(2-methoxyethyl)-4-(3-methyl-5-propyl-1-benzofuran-2-carbonyl)piperazine
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(2-oxo-1,2-dihydroquinolin-1-yl)acetamide
2-(propan-2-yl)-4-{[4-(thiophen-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyrimidine