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N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide
3-{5-[(5-cyclopropyl-4-phenyl-1H-imidazol-1-yl)methyl]-1,2-oxazol-3-yl}pyridine
(1S,5R)-6-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-[(3-fluoro-4-methoxyphenyl)methyl]-2-(pyrrolidin-1-ylmethyl)piperidine
1-[4-(pyridin-3-yl)piperazin-1-yl]-3-[5-(thiophen-2-yl)furan-2-yl]propan-1-one
4-[1-(2,4-dichlorophenyl)-1H-1,2,4-triazol-5-yl]-1-(2-methoxyethyl)pyrrolidin-2-one
2-amino-6-(furan-2-yl)-4-[2-(1H-pyrazol-1-ylmethyl)phenyl]pyridine-3-carbonitrile
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
(4aS,8aR)-6-(dimethyl-1,2-oxazole-4-carbonyl)-1-[3-(1H-imidazol-1-yl)propyl]-decahydro-1,6-naphthyridin-2-one
4-(pyridin-3-yl)-N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}pyrimidin-2-amine
N-cyclopentyl-6-{4-[1-(dimethylamino)ethyl]phenyl}pyridazin-3-amine
1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-(3-fluorophenyl)-4-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1H-pyrazole
9-(but-3-yn-1-yloxy)-4-cyclobutanecarbonyl-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-amino-6-(3,4-difluorophenyl)-4-(3-fluoro-4-hydroxy-5-methoxyphenyl)pyridine-3-carbonitrile
5-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-ylmethyl]-1,2,4-oxadiazole-3-carboxamide
1-ethyl-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-{2-[4-(6-methylpyridin-2-yl)piperazine-1-carbonyl]phenyl}morpholine
3-(2-fluorophenyl)-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
1-(3-phenyl-1H-pyrazole-4-carbonyl)-3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
1-{[4-(2-fluorophenyl)phenyl]methyl}-3-(methoxymethyl)pyrrolidine
2-{[4-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridine
N,2,5-trimethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}furan-3-carboxamide
7-[2-(4-fluorophenoxy)ethyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-(2-hydroxyethyl)-3-[5-(pyridin-4-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
2-{[4-(1-propyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]methyl}morpholine
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
3-cyclopropyl-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
5-(6-chloro-2H-chromene-3-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-ethyl-5-[4-(furan-2-yl)phenyl]-1H,4H-pyrazolo[3,4-d]imidazole
5-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)-1-[(3-methoxyphenyl)methyl]piperidin-2-one
(1S,6R)-3-[(3-methylquinoxalin-2-yl)methyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
methyl 2-(7-chloro-3-{[4-(4-ethylpiperazin-1-yl)piperidin-1-yl]methyl}-2-oxo-1,2-dihydroquinolin-1-yl)acetate
(3S,4R)-1-(2,3-dimethoxybenzoyl)-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
2-methyl-5-(4-{[3-(pyrimidin-2-yloxy)phenyl]methyl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
8-[(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2,7,8-trimethyl-N-[1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]quinoline-4-carboxamide
1-methyl-8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 1-[(4-methoxyphenyl)methyl]-5-(1H-pyrazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-2,1,3-benzothiadiazole
benzyl({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
6-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}quinoxaline
2-(2,4-difluorophenyl)-1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-(2,2-dimethyloxan-4-yl)-6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxylic acid
1-[2-(2-chlorophenyl)ethyl]-2-(methoxymethyl)-N,6-dimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
(2S,4R)-1-[(4-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-[(naphthalen-1-ylmethyl)amino]pyrrolidine-2-carboxamide
1-(3-ethyl-1H-pyrazole-4-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
2-(4-fluorophenoxymethyl)-N-methyl-N-[(4-methylphenyl)methyl]-1,3-oxazole-4-carboxamide
[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]amine