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1-[(3-fluoro-2-methylphenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-{1-[(3-chloro-4-ethoxyphenyl)methyl]pyrrolidin-3-yl}piperidine
2-amino-6-(1-methyl-1H-pyrrol-2-yl)-4-[3-(1H-pyrazol-1-yl)phenyl]pyridine-3-carbonitrile
5-{[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-N-methylfuran-2-carboxamide
6-chloro-8-methyl-3-[1-(1H-1,2,4-triazol-5-yl)ethyl]-3,4-dihydroquinazolin-4-one
4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-8-methyl-7-(pyrrolidin-1-yl)-1,2,3,4-tetrahydroquinolin-2-one
4-[(1-acetylpiperidin-4-yl)amino]-1-(2-phenylethyl)pyrrolidin-2-one
[5-({3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)furan-2-yl]methanol
2-{4-[4-(pyridin-4-yl)piperazine-1-carbonyl]piperidin-1-yl}ethan-1-ol
5-(1-methyl-1H-1,2,3-benzotriazol-5-yl)-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
5-{2-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
4-chloro-1-methyl-3-[1-(1-methylpiperidin-3-yl)-1H-imidazol-2-yl]-1H-indazole
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-7-[(2R)-oxolane-2-carbonyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[2-(2,3-dimethylphenoxy)ethyl]-1,2-dihydroquinolin-2-one
9-ethyl-1-methyl-4-[(4-methylnaphthalen-1-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(3-{[2-(3-fluorophenyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pent-4-en-1-one
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2,3,5-trimethyl-6-[3-methyl-1-(2-methylphenyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]pyrazine
2-{2-[(2-methyl-5-oxo-1,4-diazepan-1-yl)methyl]-4-(pyridin-2-yl)phenoxy}acetic acid
(2E)-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)-3-(pyridin-4-yl)prop-2-enamide
4-[4-({[1-(morpholin-4-yl)cyclopentyl]methyl}amino)piperidin-1-yl]-N-[(3S)-2-oxoazepan-3-yl]benzamide
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[2-(1H-pyrrol-1-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
6-[3-(1H-pyrazol-5-yl)phenyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-2-(2-methyl-1H-1,3-benzodiazol-5-yl)acetamide
N-[(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,4,5-trifluorobenzamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
methyl 6-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}pyrimidine-4-carboxylate
4-[2,5-dimethyl-3-(4-phenyl-1H-imidazol-5-yl)-1H-pyrrol-1-yl]-4H-1,2,4-triazole
2-butyl-N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-1,3-benzoxazole-5-carboxamide
7-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(4-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}morpholin-3-yl)acetic acid
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]acetamide
1-(1-ethylpiperidine-4-carbonyl)-4-(1-methyl-1H-imidazol-2-yl)piperidine
2-(morpholin-4-yl)-1-[4-(2-phenoxyethyl)piperazin-1-yl]butan-1-one
3,3,3-trifluoro-2-hydroxy-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}propanamide
N-[2-(dimethylsulfamoyl)ethyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
3-(methylsulfanyl)-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
N-ethyl-2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyridine-4-carboxamide
4-oxo-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
3-({[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}methyl)-7-methoxy-1,2-dihydroquinolin-2-one
methyl({[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-(3-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)acetamide
(1S,5R)-6-(pyridin-2-ylmethyl)-3-(2,2,3,3-tetramethylcyclopropanecarbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,2-dimethyl-2-(thiophen-2-ylformamido)propanamide
4-[3-(2-ethoxyethoxy)benzoyl]-2-ethyl-1-(propan-2-yl)piperazine
1-{2-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-oxoethyl}-2-methyl-1,4-dihydroquinolin-4-one
(3S,4S)-1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]piperidine-3,4-diol
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carboxamide
2-[(1-cyclopentanecarbonylpiperidin-4-yl)formamido]-2-(4-methylphenyl)acetic acid