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4-(5-methylpyridin-2-yl)-1-(5-propyl-1,3,4-oxadiazole-2-carbonyl)piperidin-4-ol
1-[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-3-carbonyl]-3-(1H-pyrazol-5-yl)piperidine
2-(1-methyl-1H-pyrrol-3-yl)-N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]acetamide
1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-phenylethane-1,2-dione
[(3R,4S)-4-[(4-ethylpiperazin-1-yl)methyl]-1-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl]methanol
1-(5-ethyl-1,3-oxazole-4-carbonyl)-4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
6-{2-amino-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}-1H,2H,3H,4H,5H,6H,7H,8H-pyrazolo[3,4-d]azepin-3-one
N-[(3S,4R)-1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
1-(2-methoxybenzoyl)-4-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]piperazine
3-(3,4-dimethylphenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]propan-1-one
(2S,4R)-1-[(4-hydroxy-3,5-dimethoxyphenyl)methyl]-N-(propan-2-yl)-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
1-benzyl-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
[(3R,5R)-5-(morpholin-4-ylmethyl)-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl]methanol
methyl 4-{[4-(oxan-2-ylmethoxy)phenyl]carbamoyl}piperazine-1-carboxylate
1-[(1S,5R)-6-(1-benzothiophene-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
(2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-(morpholine-4-carbonyl)pyrrolidine-2-carboxylic acid
(2E)-3-(2-chlorophenyl)-N-[(3,4-dimethoxyphenyl)methyl]-N-(pyridin-2-ylmethyl)prop-2-enamide
(2E)-1-[4-(3-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}phenoxy)piperidin-1-yl]-3-(4-methoxyphenyl)prop-2-en-1-one
7-[(2,3-difluorophenyl)methyl]-2-(pyrazin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[(3-chlorophenyl)methyl]-N,2-dimethyl-6-(piperidin-4-yl)pyrimidin-4-amine
3-[2-(2,6-difluorophenyl)ethyl]-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidine
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-(4-methyl-1H-imidazol-1-yl)acetamide
1-[4-(4-fluorophenyl)oxane-4-carbonyl]-4-hydroxypiperidine-4-carboxylic acid
N2-(1,4-dioxan-2-ylmethyl)-N4-ethyl-N2-methylpyrimidine-2,4-diamine
N-cyclopentyl-1-{1-[(4-ethylphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
(3R,4S)-3,4-dimethyl-1-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}piperidin-4-ol
(3R,5S)-1-benzyl-N3-(4-fluorophenyl)-N5-(oxolan-2-ylmethyl)piperidine-3,5-dicarboxamide
5-fluoro-N-[1-(1,3-thiazol-5-yl)propan-2-yl]quinazolin-4-amine
(2R,6R)-6-methyl-1-{[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]methyl}-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
5-[3-(4-ethoxy-3-methylphenyl)propyl]-1-methyl-1H-1,2,4-triazole
N-(2-{1-[3-(2,4-difluorophenyl)propanoyl]piperidin-2-yl}ethyl)acetamide
N-[3-(2-methoxyethoxy)phenyl]-2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidine-1-carboxamide
2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-4-(2,4-dioxoimidazolidin-1-yl)benzamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(3,3,3-trifluoropropyl)pyrrolidine-3-carboxylic acid
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxamide
N-[2-(4-chlorophenyl)-2-(pyrrolidin-1-yl)ethyl]-3-ethyl-4-methyl-1H-pyrazole-5-carboxamide
methyl 3-[1-(4-methyl-1H-imidazole-5-carbonyl)piperidin-2-yl]propanoate
6-{[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]sulfonyl}-4-methylquinolin-2-ol
ethyl 2-{4-[(3-methoxyphenyl)methyl]-3-oxopiperazin-1-yl}-1,3-oxazole-4-carboxylate
2-[5-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)-1-(3,5-dimethylphenyl)-1H-1,2,4-triazol-3-yl]acetamide
N-[2-(benzyloxy)ethyl]-4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
3-(4-phenylbenzoyl)-1-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]piperidine
N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
2-[3-(2-methylphenyl)-1H-pyrazol-1-yl]-N-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]acetamide
1-cyclobutanecarbonyl-N-[1-(pyrimidin-2-yl)piperidin-3-yl]piperidine-4-carboxamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N,N-dipropyl-1,3-oxazole-4-carboxamide
(4aS,8aR)-1-butyl-6-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
7-[4-(3-hydroxy-3-methylbutyl)benzoyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one