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(4aS,7aR)-1-(2-aminopyridine-4-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-4-(morpholin-4-yl)butan-1-one
(1R,5R)-6-(cyclobutylmethyl)-3-(4-propyl-1,2,3-thiadiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carboxamide
1-methyl-N-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-N-(pyridin-3-ylmethyl)piperidin-4-amine
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-1,4-dithiepan-6-amine
4-{4-[1-(1H-indazol-6-yl)-1H-imidazol-2-yl]phenyl}but-3-yn-1-ol
4-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-1-(1-methylpiperidin-4-yl)piperidine
N-[3-(dimethylamino)-2,2-dimethylpropyl]-1-ethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-3-(4-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
1-{[3-(cyclopentyloxy)phenyl]methyl}-4-(pyridin-3-ylmethyl)piperazine
N-{1-[1-(2-fluorophenyl)-1H-1,2,4-triazol-5-yl]ethyl}propanamide
1-[7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-(1H-indazol-1-yl)ethan-1-one
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]-1,4-diazepan-5-one
N-[2-(2-fluorophenyl)-1-[1-(quinolin-6-ylmethyl)piperidin-4-yl]ethyl]-N-methylthiophene-3-carboxamide
1-[(3-methylphenyl)methyl]-4-[3-(1-methylpiperidin-3-yl)propanoyl]piperazin-2-one
3-[(1-benzyl-1H-imidazol-5-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2S)-2-[3-(azocan-1-yl)propanamido]-3-phenylpropanoic acid
(3S,9aR)-8-(4-chlorobenzoyl)-2-methyl-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-{5-[(2-methyl-1,3-thiazol-4-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
2-chloro-4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]phenol
4-cyclopropyl-1-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-4-methylpyrrolidin-2-one
7-(3-methoxyphenyl)-2-(2-methyl-1,3-thiazol-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-{[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]methyl}-1-methyl-1,2-dihydroquinolin-2-one
4-{[4-(benzyloxy)piperidin-1-yl]methyl}-2-methoxyphenol
2-{2-[2-fluoro-6-(propan-2-yloxy)phenyl]phenyl}-5-methyl-1,3,4-oxadiazole
1-(6-hydroxy-1,4-oxazepan-4-yl)-2-(2-phenylindolizin-3-yl)ethane-1,2-dione
(4aS,8aR)-1-(2-aminoethyl)-6-(5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-[(4-fluorophenyl)methyl]acetamide
ethyl 4-[(4-chlorophenyl)methyl]piperidine-4-carboxylate
2-[(6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridazin-3-yl)amino]ethan-1-ol
2-amino-N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-4-phenylpyrimidine-5-carboxamide
(2R,3S,6R)-3-(3-methoxyphenyl)-5-[(5-methylfuran-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
3-acetamido-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)benzamide
[(4,5-dimethylfuran-2-yl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)methylamine
2-({1-[(2,5-dimethylphenyl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
2-methyl-N-[3-(3-phenylpropanamido)phenyl]-1H-imidazole-4-carboxamide
3-(1H-imidazol-1-ylmethyl)-1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperidine
1-[5-(1-cyclohexylpiperidin-4-yl)-3-methyl-1H-1,2,4-triazol-1-yl]butan-2-ol
1-(2-chloroprop-2-en-1-yl)-3-{[(2,3-dihydroxypropyl)amino]methyl}-6,7-dimethoxy-1,2-dihydroquinolin-2-one
1'-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
ethyl 5-(2,2-diphenylethyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(cyclopropylmethyl)-N-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
3-methoxy-5-(4-phenyl-1H-imidazol-1-yl)pyridine
1-[(dimethyl-1,3-thiazol-5-yl)methyl]-4-[(4-fluorophenyl)methyl]piperidine
3-[1-(5-cyclopropyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-N-[(5-methylfuran-2-yl)methyl]propanamide
4-[(1-methyl-1H-pyrrol-2-yl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{4-[(2-butyl-1H-imidazol-4-yl)methyl]-1-cyclopentylpiperazin-2-yl}ethan-1-ol
2-(2-{[(butan-2-yl)(pyridin-4-ylmethyl)amino]methyl}phenoxy)ethan-1-ol