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2-cyclopropyl-9-[2-(methylamino)acetyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-[3-(cyclopentylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N-ethylpyrimidin-4-amine
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-cyclopropyl-1H-1,2,4-triazole
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)acetamide
3-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-1-[4-(oxolan-2-ylmethoxy)phenyl]urea
2-amino-4-[2-(difluoromethoxy)phenyl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-(2,3-dihydro-1H-inden-2-yl)-N-[3-(furan-2-yl)phenyl]piperidine-4-carboxamide
3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-(1,2,3,4-tetrahydronaphthalen-1-yl)propanamide
6-(2,3-dihydro-1-benzofuran-7-yl)-N,N-dimethylpyridine-2-carboxamide
4-methyl-2-(propan-2-yl)-N-propyl-N-(thiophen-3-ylmethyl)-1,3-thiazole-5-carboxamide
2-(3-{1-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrazol-3-yl}phenyl)benzonitrile
N-[1-(1H-indol-2-yl)ethyl]-N,2,4-trimethyl-1,3-thiazole-5-carboxamide
8-[(2-aminopyridin-3-yl)methyl]-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[5-fluoro-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-methyl-1H-indol-3-yl)acetamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)quinoxalin-2-amine
2-(4,5-dimethyl-1H-imidazol-1-yl)-1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
3-{1-[1-(thiolan-3-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}pyridine
ethyl({[2-(prop-2-en-1-yloxy)phenyl]methyl}){[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
4-[2-({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amino)ethyl]phenol
dimethyl({5-[2-(2-phenylethyl)morpholine-4-carbonyl]furan-2-yl}methyl)amine
N-cyclohexyl-N,4-dimethyl-5-(1-{[(4-methyl-1H-imidazol-2-yl)methyl]amino}ethyl)pyrimidin-2-amine
4-[3-(4-fluorophenoxy)propyl]-1,3λ6,4-oxathiazinane-3,3-dione
2-[5-(1,5-dimethyl-1H-pyrrol-2-yl)-3-phenyl-1H-1,2,4-triazol-1-yl]ethan-1-ol
4-ethyl-1-methyl-3-[1-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(2-aminoethyl)-N-[2-methyl-1-(pyrrolidin-1-yl)propan-2-yl]quinazolin-4-amine
1-{4-[(4-fluoro-3-methoxyphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-9-yl}butan-1-one
2-[(7-methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)amino]-N-(propan-2-yl)acetamide
3-methoxy-2-[3-(morpholin-4-ylmethyl)phenyl]pyridin-4-amine
3-{[methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amino]methyl}phenol
N-(4-fluoro-2-methylphenyl)-3-{1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidin-3-yl}propanamide
N-{1-[7-(2,5-dimethylfuran-3-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-2-methylpropyl}pyridine-2-carboxamide
2-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]-8-methyl-2,8-diazaspiro[4.5]decane
4-({[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]carbamoyl}amino)-N-(2-methoxyethyl)-3-methylbenzamide
2-(2,5-dioxoimidazolidin-1-yl)-N-[2-phenyl-2-(piperidin-1-yl)ethyl]acetamide
N-(2,3-dihydro-1H-inden-1-yl)-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-[(3S,4R)-4-(4-methylphenyl)-1-[3-(pyridin-2-yl)propanoyl]pyrrolidin-3-yl]acetamide
(2S)-2-amino-N-propyl-N-(pyridin-3-ylmethyl)-3-(1,3-thiazol-4-yl)propanamide
4-ethyl-5-({5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1,3-thiazol-2-amine
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
5-{[2-(4-ethylphenyl)-1H-imidazol-1-yl]methyl}-3-(propan-2-yl)-1,2,4-oxadiazole
4-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-4-oxobutane-1-sulfonamide
(3S,4S)-4-[(dimethylamino)methyl]-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-3-ol
1-({[(4-{3-[benzyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]amino}methyl)cyclohexan-1-ol
5-propyl-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)pyrimidin-4-amine
1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
methyl({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)[2-(pyridin-2-yl)ethyl]amine
5-{2-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperidine-3-carboxamide
[3-benzyl-1-(3-methylthiophene-2-carbonyl)piperidin-3-yl]methanol
1-benzyl-5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide