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2-[3-(2-cyclopropyl-1H-imidazol-1-yl)phenyl]pyridine
7-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-{1-[(3-chloro-4,5-diethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
5-[1-(furan-3-ylmethyl)pyrrolidin-2-yl]-N-(1-methyl-1H-pyrazol-5-yl)thiophene-2-carboxamide
4-ethyl-N-(2-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}-2-oxoethyl)cyclohexane-1-carboxamide
3-{[1-ethyl-3-(hydroxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyrrolidin-3-ol
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-3-cyclopropyl-1H-pyrazole-5-carboxamide
1-(4-methylpentanoyl)-4-(2-methylpropyl)-1,4-diazepan-5-one
methyl(oxan-2-ylmethyl){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
5-methyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-1-propyl-1H-pyrazole-4-carboxamide
1-(2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-oxoethyl)azepan-2-one
2-[3-(2-methylphenyl)benzoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-[(4-methoxypyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(4aR,7aS)-1-acetyl-4-(3-chloro-4-methoxybenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-ethyl-5-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-1H-indole
2-(1H-imidazole-4-carbonyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
(3R)-3-[1-(2-methoxyphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydroisoquinoline
5-{[7-(2-hydroxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]methyl}-N-methyl-1,2,4-oxadiazole-3-carboxamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-phenylpropanamide
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-4-(pyridin-2-yl)pyrimidin-2-amine
2-[3-(methylsulfanyl)propanoyl]-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
1-[(2-aminopyridin-3-yl)methyl]-4-(oxan-4-yl)-1,4-diazepan-6-ol
2-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidine-1-carbonyl]benzonitrile
N-[2-(2-ethylphenoxy)ethyl]-3-(4-hydroxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
2-{2-[(3-hydroxy-3-phenylpyrrolidin-1-yl)methyl]phenoxy}acetic acid
7-[(4-methyl-1H-imidazol-5-yl)methyl]-N-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-ethyl-N-(oxan-4-ylmethyl)-2-{[(2E)-3-phenylprop-2-en-1-yl]sulfanyl}pyridine-3-carboxamide
4-(1-hydroxy-3-methylbutyl)-N-(3-phenyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-[(1-ethylpiperidin-4-yl)amino]-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
N-[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]-2-(4-methyl-1,4-diazepan-1-yl)acetamide
N-(5-tert-butyl-2-methoxyphenyl)-2-(hydroxymethyl)azepane-1-carboxamide
N-[(3R,4R)-1-[(2,4-dimethoxyphenyl)methyl]-3-hydroxypiperidin-4-yl]pyridine-3-carboxamide
N-{[4-(6-methoxypyridin-3-yl)phenyl]methyl}cyclopropanamine
1-(3-chlorophenyl)-4-[1-(3-methylthiophene-2-carbonyl)piperidin-3-yl]piperazine
5-ethyl-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1H-pyrrole-2-carboxamide
({5-[(4-chlorophenyl)sulfanyl]furan-2-yl}methyl)[2-(1H-imidazol-4-yl)ethyl]amine
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-2-fluoro-5-sulfamoylbenzamide
N-(pyridin-2-ylmethyl)-5-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
7-(3,6-dimethylpyrazin-2-yl)-4-(1-methylpiperidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(3-chlorophenyl)-5-methyl-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperazin-2-one
1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(piperidin-1-yl)ethan-1-one
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
(3S,4R)-1-(3-carboxybenzoyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-(2-methoxyethyl)-1-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
N-(1-{5-[(cyclohexylmethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)-2-(2-methyl-1,3-thiazol-4-yl)acetamide
4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-N-(propan-2-yl)pyridine-2-carboxamide
2-(4-{[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]sulfonyl}phenoxy)acetamide
2-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
(1S,5R)-3-[(5-chloro-2,3-dimethoxyphenyl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
(2R,3R)-3-amino-1'-(pyridin-2-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol