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4-[4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazol-3-yl]-1-methylpyrrolidin-2-one
(3-{[(2H-1,3-benzodioxol-5-ylmethyl)(pyridin-3-ylmethyl)amino]methyl}-2,4,6-trimethylphenyl)methanol
(4aS,8aR)-1-(3-methoxypropyl)-6-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-{thieno[2,3-d]pyrimidin-4-yl}piperidine
1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-2-(quinazolin-4-yloxy)ethan-1-one
{4-[5-(3-chloropyridin-4-yl)-1,2,4-oxadiazol-3-yl]phenyl}methanol
(2S)-N-[4-(3-methoxyphenyl)phenyl]-1-(1,3-oxazole-5-carbonyl)pyrrolidine-2-carboxamide
2-chloro-N-[2-(3-methoxypropanoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
(1S,3R)-3-amino-N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}cyclopentane-1-carboxamide
N'-(3-chloro-4-fluorophenyl)-N-(furan-2-ylmethyl)-N-(prop-2-yn-1-yl)butanediamide
3,3,3-trifluoro-N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}propanamide
3,8-bis(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}-5-phenylpyrazolo[1,5-a]pyrimidine
4-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-1-methylimidazolidin-2-one
1-amino-N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]cyclopropane-1-carboxamide
3-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-1-[2-methyl-4-(pyrrolidine-1-carbonyl)phenyl]urea
(3S,4R)-1-[(3,5-dimethoxyphenyl)methyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
7-(5-chloropyridin-2-yl)-4-(cyclobutylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
8-(3-methyl-1,2-oxazole-5-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-ethyl-2-(3-hydroxypiperidin-1-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
N-[(3,4-difluorophenyl)methyl]-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-methyl-5-{4-[(8-methylquinolin-5-yl)methyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxamide
3-[(3R,4S)-1-[(3-methylquinoxalin-2-yl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
5-butyl-4-(1H-pyrazole-3-carbonyl)-1-(5,6,7,8-tetrahydronaphthalen-1-yl)piperazin-2-one
N-[2-(1-benzylpyrrolidin-3-yl)ethyl]-1-ethyl-3-methyl-1H-pyrazole-4-carboxamide
4-(carbamoylmethoxy)-2-hydroxy-5-[(1E)-pent-1-en-1-yl]benzoic acid
3-{2-[1-(2-methyl-1,3-benzothiazol-6-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,4-triazol-5-amine
9-(2-methoxy-3-methylbenzoyl)-3-oxa-9-azaspiro[5.5]undecane
N,N-dimethyl-2-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine-3-carboxamide
{1-ethyl-5-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-[2-(4-methoxyphenyl)ethyl]piperidin-2-one
{5-[4-(2-methylphenoxy)piperidine-1-carbonyl]-1H-1,3-benzodiazol-2-yl}methanol
3-(3,4-difluorophenyl)-1-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]propan-1-one
(4aS,8aS)-2-cyclopentanecarbonyl-7-(1-methyl-1H-pyrazole-4-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
1-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
1-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-2-methyl-1,4-diazepan-5-one
1-[(4-chlorophenyl)methyl]-N-methyl-N-[(5-methylfuran-2-yl)methyl]-6-oxopiperidine-3-carboxamide
3-butyl-4-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1-methylpiperazin-2-one
1-methyl-N-({2-[(2-oxopyrrolidin-1-yl)methyl]phenyl}methyl)azepane-2-carboxamide
5-chloro-4,6-dimethyl-3-[4-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
3-{[(1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
2-(1,4-dimethylpiperazin-2-yl)-1-[4-(hydroxymethyl)-4-(2-phenylethyl)piperidin-1-yl]ethan-1-one
3-(2-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,2,3-oxadiazol-3-ium-5-olate
4-(4-methylpyridine-3-carbonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-2-(2-oxopyrrolidin-1-yl)propanamide
1-ethyl-3-(naphthalen-1-ylmethyl)-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(4-chloro-1H-pyrazol-1-yl)-1-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]propan-1-one
1-[(8-fluoroquinolin-2-yl)methyl]-1,4-diazepane-6-carboxylic acid