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1-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}-2-[4-(dimethylamino)phenyl]ethan-1-one
1-(3-carbamoylpyridin-2-yl)-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
5-({[(1-hydroxycyclohexyl)methyl]carbamoyl}amino)-2-methoxy-N,N-dimethylbenzamide
1-(2,3-dihydro-1H-inden-2-yl)-4-{[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]amino}pyrrolidin-2-one
N,3-dimethyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}furan-2-carboxamide
(4aS,7aR)-1-{6-chloro-2-methylimidazo[1,2-a]pyridine-3-carbonyl}-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{5-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-1H-pyrazol-3-yl}ethan-1-one
N-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-N-(pyridin-2-ylmethyl)cyclohexanamine
2-tert-butyl-1-[3-(1H-imidazol-1-yl)propyl]-1H-imidazole
8-(2-cyclopropylacetyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-N-[(4-fluorophenyl)methyl]propanamide
1-[3-(3-benzyl-1H-1,2,4-triazol-5-yl)propyl]piperidin-2-one
methyl 6-(5-methyl-1H-indol-3-yl)pyridine-3-carboxylate
N-ethyl-6-[3-(2-hydroxyethyl)-4-(thiophen-3-ylmethyl)piperazin-1-yl]pyridine-3-carboxamide
(4-methyl-5-{1-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-3-yl}-4H-1,2,4-triazol-3-yl)methanol
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-2H-1,3-benzodioxole-5-carboxamide
8-{5-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl}quinoline
4-(naphthalen-2-yloxy)-1-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxylic acid
1-benzoyl-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-{5-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
[(3R,4R)-4-[(dimethylamino)methyl]-1-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}pyrrolidin-3-yl]methanol
methyl 2-[(2-methylpropyl)sulfamoyl]-6-{2-[4-(methylsulfanyl)phenyl]acetyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(4-methoxy-2-methylphenyl)-2-[4-(propan-2-yl)piperazin-1-yl]acetic acid
6-cyclopentyl-N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N,1-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3R,4R)-1-{[5-(2-methylpropyl)thiophen-2-yl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
2-ethyl-4-phenyl-9-(pyridine-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
3-ethyl-1-[4-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-3-[2-(1H-pyrazol-1-yl)ethyl]urea
2-cyclobutyl-N-(2,3-dihydro-1H-inden-2-yl)-1-methyl-7-(oxolane-2-amido)-1H-1,3-benzodiazole-5-carboxamide
2-(pyridin-4-ylmethyl)-8-(1,3-thiazol-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
8-({2-[2-(4-methylpiperazin-1-yl)ethoxy]phenyl}methyl)-2,8-diazaspiro[4.5]decan-3-one
5-{1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]pyrrolidin-2-yl}-N-methylthiophene-2-carboxamide
N-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-2-[methyl(pyridin-4-ylmethyl)amino]acetamide
5-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
6-{4-[2-(dimethylamino)-2-(3-fluorophenyl)acetyl]piperazin-1-yl}pyridine-3-carbonitrile
1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-4-(5-ethylfuran-2-yl)-1H-1,2,3-triazole
7-fluoro-2-[4-(furan-3-carbonyl)-1,4-diazepane-1-carbonyl]-3-methyl-1H-indole
propan-2-yl 3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxylate
1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(pyridin-2-yl)piperazine
dimethyl(3-{2-[1-(3-methyl-1,2-oxazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
(3S,4R)-1-(3-methanesulfonylbenzoyl)-3-methoxypiperidin-4-amine
4-{4-[1-(cyclohexylmethyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}butanamide
N-[1-(1,3-thiazol-5-yl)propan-2-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
2-[1-(1-methylpiperidin-4-yl)-4-[(3-methylthiophen-2-yl)methyl]piperazin-2-yl]ethan-1-ol
5-[4-(2-chlorophenyl)piperazine-1-carbonyl]-N-(cyclohexylmethyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
4-{1-[3-(methylsulfanyl)propyl]-4-phenyl-1H-imidazol-5-yl}pyridine
5-[({[3-(2-{4-[(2E)-3-(3-fluorophenyl)prop-2-enoyl]piperazin-1-yl}ethoxy)phenyl]methyl}(methyl)amino)methyl]pyrrolidin-2-one
N-(3-chloro-4-fluorophenyl)-3-{1-[(4-acetamidophenyl)methyl]piperidin-4-yl}propanamide
1-(2,4-dimethylphenoxy)-3-{[4-(methylsulfanyl)butan-2-yl]amino}propan-2-ol
2-{3-[1-(2-methylphenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]piperidin-1-yl}acetamide
4-cyano-N-ethyl-1-methyl-N-(pyridin-4-ylmethyl)-1H-pyrrole-2-carboxamide