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7-{[2-(pyridin-3-yl)piperidin-1-yl]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
4-{[2-(1-benzofuran-5-yl)phenyl]methyl}morpholine
1-methyl-5-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
N-benzyl-N-(2-hydroxyethyl)-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
5-(3-methoxyphenoxymethyl)-N-(1H-1,2,4-triazol-3-ylmethyl)-1H-pyrazole-3-carboxamide
(3R,4R)-1-[1-(4-fluoro-2-methylphenyl)piperidin-4-yl]-3,4-dimethylpyrrolidin-3-ol
N-(2-phenylethyl)-3-(1H-1,2,3,4-tetrazol-1-yl)-5-(2,3,4-trimethoxyphenyl)benzamide
2-[(5-{[butyl(furan-2-ylmethyl)amino]methyl}pyrimidin-2-yl)amino]acetic acid
N,N-dimethyl-2-{[2-(pyridin-2-ylsulfanyl)acetamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-{1'-[2-(morpholin-4-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
3-cyclohexyl-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-1H-pyrazole-4-carboxamide
2-(diethylamino)-1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-(pyrrolidin-3-yl)benzamide
1-[(2,4-difluoro-3-methoxyphenyl)methyl]-N-methylpiperidine-2-carboxamide
2-(4-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}phenyl)acetamide
N3-cyclooctyl-N5-[(3-methoxyphenyl)methyl]-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
3-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}-8-methyl-2-(thiophen-2-yl)quinoline
2-[2-(dimethylamino)ethyl]-9-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[(2R)-oxolane-2-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-4-methylpyrimidine-5-carboxamide
9-(1-methyl-1H-pyrazole-3-carbonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(1-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}piperidin-4-yl)-3-(pyrrolidine-1-carbonyl)piperidine
4-(1-benzothiophen-2-ylmethyl)piperazine-1-sulfonamide
N-{[2-(4-acetylpiperazin-1-yl)-6-methylquinolin-3-yl]methyl}-N-[2-(cyclohex-1-en-1-yl)ethyl]furan-3-carboxamide
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-3-(pyridin-3-yl)propanamide
5-[({[1-(2-methoxyethyl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)amino)methyl]-N,N-dimethyl-1,3-thiazol-2-amine
2-[(2-methoxypyridin-3-yl)methyl]-2,3-dihydro-1,2-benzothiazol-3-one
N-(cyclobutylmethyl)-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
[(2S)-1-{2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzoyl}pyrrolidin-2-yl]methanol
(3R,4S)-4-[4-(8-fluoroquinoline-2-carbonyl)-1,4-diazepan-1-yl]oxolan-3-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-ethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{[2-(4-chlorophenyl)-7-methoxyquinolin-3-yl]methyl}piperidin-4-ol
N-[5-({7-[ethoxy(phenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}methyl)thiophen-2-yl]acetamide
4-[(2,4-dichlorophenyl)methyl]-3-[2-(1H-pyrazol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(3aR,6aR)-2-methanesulfonyl-5-(2-methylpyrimidin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-methyl-N-[2-({1-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]piperidin-4-yl}amino)ethyl]methanesulfonamide
(2R,6R)-11-methoxy-4-(4-methyl-1,3-thiazole-5-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-[2-(cyclohexylsulfanyl)ethyl]-3-(4-methanesulfonylphenyl)urea
3-{5-[3-(4-fluorophenoxy)propyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
1-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-N-(1H-pyrazol-3-ylmethyl)piperidin-4-amine
1-(2-chloropyridin-3-yl)-3-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]urea
5-ethyl-N-[1-(4-methanesulfonylphenyl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
5-(5-chloro-2-hydroxybenzoyl)-N-(2-hydroxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-(2-methylphenoxy)-1-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}azetidine
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(3-methylpiperidin-1-yl)methyl]phenoxy]-N-(5-fluoro-2-methylphenyl)acetamide
7-(2-methoxyphenyl)-2-{[(1-methyl-1H-imidazol-2-yl)sulfanyl]methyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}-2-(pyrrolidin-1-yl)ethan-1-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-(4-methylphenyl)-1H-pyrazole-5-carboxamide
5-{[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
5-methoxy-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]furan-2-carboxamide