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3-[4-(1-benzyl-3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]-1λ6-thiolane-1,1-dione
1'-(1-benzofuran-5-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(3S,4R)-4-(2-methylphenyl)-1-(quinoxaline-6-carbonyl)pyrrolidine-3-carboxylic acid
N,N-dimethyl-2-[methyl({[2-(pyridin-2-yl)pyrimidin-5-yl]methyl})amino]propanamide
N-[1-(3-methylphenyl)-5-oxopyrrolidin-3-yl]-4-(piperidin-1-ylmethyl)benzamide
2-(4-{1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl}piperidin-1-yl)pyrimidine
3-{2,7-diazaspiro[4.5]decane-2-sulfonyl}-N-methylbenzamide
2-[2-(aminomethyl)-7-fluoro-2,3-dihydro-1-benzofuran-5-yl]quinoline-4-carboxylic acid
4-{[1-(2,3-dihydro-1H-inden-2-yl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}morpholine
1-methyl-3-(5-propyl-4H-1,2,4-triazol-3-yl)-1-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}urea
(3S,4R)-1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
7-[(4-fluorophenyl)methyl]-2-(furan-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-({1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
(3-{2-azabicyclo[2.2.1]hept-5-en-2-yl}propyl)({[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl})amine
2-(4-chloro-1H-pyrazol-1-yl)-N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}acetamide
(1-{2-[(1-benzoylpiperidin-4-yl)amino]ethyl}piperidin-2-yl)methanol
2-(4-methanesulfonylphenyl)-1-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
2-(morpholin-4-yl)-N-[(2-phenoxypyridin-3-yl)methyl]butanamide
N5-[(4-methoxyphenyl)methyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-ethyl-N-[(3-methylpyridin-2-yl)methyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-[2-(1H-indol-1-yl)ethyl]-N-methylbenzamide
[(3R,5R)-1-(2-benzyl-1,3-thiazole-4-carbonyl)-5-[(dimethylamino)methyl]piperidin-3-yl]methanol
1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-2-{methyl[(4-methylphenyl)methyl]amino}ethan-1-one
3,3-dimethyl-1-({5-[(5-methylnaphthalen-1-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)urea
2-(methylsulfanyl)-4-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
N-{2-[3-(ethylsulfanyl)-5-oxo-4,5-dihydro-1,2,4-triazin-6-yl]phenyl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
2-(4-chloro-2-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1H-imidazol-2-yl}phenoxy)acetamide
1-(4-cyclobutanecarbonyl-1,4-diazepan-1-yl)-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
(4aR,8aS)-1-(2-cyclopentylacetyl)-N,N-dimethyl-decahydro-1,6-naphthyridine-6-sulfonamide
(3aS,6aR)-5-(5-methylpyrazine-2-carbonyl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-4-[(1-methylpiperidin-4-yl)methyl]piperazine
9-methoxy-7-(6-methoxypyridin-2-yl)-4-(3-methylbutyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(7-methoxy-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
2-(prop-2-en-1-yl)-9-(quinoxaline-6-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
{[4-methoxy-3-(methoxymethyl)phenyl]methyl}({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl})amine
7-fluoro-2-[3-(1H-imidazol-1-yl)propyl]-4-methylquinoline
2,3-dioxo-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-ethyl-N-(2-methoxyethyl)piperidine-3-carboxamide
N4-cyclopropyl-6-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine-2,4-diamine
2-{[({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]methyl}-3,4-dihydroquinazolin-4-one
9-(3-methyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(2-aminoethyl)-N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]quinazolin-4-amine
N-[2-(4,5-dimethyl-1H-imidazol-1-yl)ethyl]-6-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
8-fluoro-3-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,4-dihydroquinolin-4-one
2-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]formamido}-4-(methylsulfanyl)butanoic acid
4-{2-[1-(2-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethyl}-3-methyl-4H-1,2,4-triazole
N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]-2-(methylamino)pyridine-3-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)acetamide
5-methyl-N-[1-(pyridin-2-yl)propan-2-yl]-1-[4-(pyridin-3-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide