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6-chloro-2-{2-oxo-2-[3-(4-phenoxybenzoyl)piperidin-1-yl]ethyl}-2,3-dihydropyridazin-3-one
6-(2-cyanophenyl)-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(2-methoxyethyl)methylamine
4-(5-chloro-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1λ6-thiomorpholine-1,1-dione
2-{1-[(2-chloro-4-fluorophenyl)methyl]piperidin-2-yl}acetic acid
8-[2-(5-chloro-6-methyl-1-benzofuran-3-yl)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
9-hydroxy-3-[4-(3-methylphenoxy)piperidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
3-(3,5-dimethyl-1H-pyrazol-1-yl)-1-(4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)propan-1-one
3-(cyclopentylsulfamoyl)-5-[4-(hydroxymethyl)phenyl]benzoic acid
7-fluoro-3-[2-(morpholin-4-yl)ethyl]-3,4-dihydroquinazolin-4-one
N4-methyl-N4-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-2-(pyrrolidin-1-yl)pyrimidine-4,6-diamine
(1R,5R)-6-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
5-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-2-(pyridin-4-yl)pyrimidine
1-[4-(3-methoxyphenyl)benzoyl]-4-(1-methyl-1H-imidazol-2-yl)piperidine
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-2-(1-methyl-1H-pyrazol-3-yl)piperidine
3-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-1-[(5-methyl-1H-pyrazol-3-yl)methyl]urea
4-{2-[2-(1-phenylethyl)-1H-imidazol-1-yl]ethyl}benzene-1-sulfonamide
2-{4-[(4-fluorophenyl)methyl]-3-oxopiperazin-1-yl}-2-(thiophen-3-yl)acetic acid
1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-2-(2H-indazol-2-yl)ethan-1-one
1-[(4aR,8aS)-1-[2-(2,3,4-trifluorophenyl)acetyl]-decahydro-1,6-naphthyridin-6-yl]-2-phenoxyethan-1-one
5-methyl-4-({1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}amino)thieno[2,3-d]pyrimidine-6-carboxylic acid
6-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidine-1-carbonyl)-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
1-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]-3-[3-(1H-1,2,3-triazol-1-yl)propyl]urea
(1R,5R)-6-[(2-fluoro-5-methoxyphenyl)methyl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-(3-benzyl-1H-1,2,4-triazol-5-yl)-1-[(4-methoxyphenyl)methyl]-1-methylurea
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]propanamide
(2E)-3-(3,4-dimethoxyphenyl)-N-[2-(4-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxy)propyl]prop-2-enamide
1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-2-(3-methoxyphenyl)azetidine
N-{[2-(2-cyclobutaneamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,3-dimethoxybenzamide
2-(5-chloro-2-methoxyphenyl)pyridine-4-carboxamide
2-(2-{5-[1-(2-methoxyethyl)piperidin-4-yl]-4-phenyl-1H-imidazol-1-yl}ethoxy)ethan-1-ol
{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]amine
N-cyclopentyl-2-phenyl-5,6,7,8-tetrahydroquinazolin-5-amine
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-[(3-ethyl-1H-pyrazol-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
3-{[(2-hydroxy-2-methylpropyl)carbamoyl]methyl}-N-(2-methoxyethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-hydroxy-1-[3-(2-methoxyphenoxy)azetidin-1-yl]-4-methylpentan-1-one
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
2,3-dimethyl-5-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]benzene-1-sulfonamide
(3R,5R)-N-[3-(dimethylamino)propyl]-1-(2-phenylethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-3-carboxamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-(methylsulfanyl)pyrimidine-5-carboxamide
(1R,3S)-3-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]cyclopentane-1-carboxylic acid
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]acetamide
5-amino-N-(2H-1,3-benzodioxol-5-ylmethyl)-N-[(4-methylphenyl)methyl]-1H-pyrazole-3-carboxamide
8-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(3,5-dichlorophenyl)-6-(hydroxymethyl)-1,4-oxazepane-4-carboxamide
1-(furan-2-carbonyl)-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine
N-[2-(dimethylamino)ethyl]-5-(4-fluoro-3-methylbenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-(4-fluorophenyl)-1-{4-[2-(3-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}phenoxy)ethyl]piperazin-1-yl}ethan-1-one
1-(3-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-6-methylquinolin-2-yl)piperidin-3-ol
N-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}phenyl)acetamide