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2-{4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-1,4-diazepan-1-yl}-1,3-benzothiazole
2-{5-[1-(3-phenyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetic acid
5-{6-amino-5-cyano-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]pyridin-2-yl}-2,4-dimethyl-1H-pyrrole-3-carboxylic acid
2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}acetamide
2-[(4-methoxyphenyl)methyl]-4-[(2-phenyl-1,3-oxazol-4-yl)methyl]morpholine
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[2-(2-oxoimidazolidin-1-yl)ethyl]pyrimidine-5-carboxamide
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-cyclopropyl-5-oxopyrrolidine-3-carboxamide
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-2-(2,3-dimethylphenoxy)-N-methylacetamide
1-[(4-methylphenyl)methyl]-4-(pyridin-4-ylmethyl)piperazin-2-one
1-(1H-imidazol-4-ylmethyl)-4-(oxolane-2-carbonyl)-1,4-diazepane
N-benzyl-2-{2-methyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}propanamide
2-(3-fluorophenoxymethyl)-N-[(3-methoxyphenyl)methyl]-1,3-oxazole-4-carboxamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(2,6-dimethylpyrimidine-4-carbonyl)pyrrolidin-3-yl]methanol
4-methoxy-2-{[9-methoxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenol
1-ethyl-N-(furan-2-ylmethyl)-N-methyl-5-[methyl(2-methylpropyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3S,9aR)-3-(cyclohexylmethyl)-8-[(4-methylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-({1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}methyl)-4-phenylbenzamide
8-[2-(2-methylphenyl)benzoyl]-1-oxa-8-azaspiro[4.5]decane
1-[2-(2-benzyl-3-oxopiperazin-1-yl)-2-oxoethyl]-1,2-dihydropyrimidin-2-one
1-methyl-N-{[5-(methylcarbamoyl)furan-2-yl]methyl}-1H-indole-6-carboxamide
1-ethyl-3-[(3-methoxyphenyl)methyl]-8-[1-(methylsulfanyl)propan-2-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(3R,4S)-1-(4-methanesulfonylbenzoyl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
(3E)-1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}hex-3-en-1-one
(2S,4S)-1-[(5-chlorothiophen-2-yl)methyl]-N-ethyl-4-(3-methoxypropanamido)pyrrolidine-2-carboxamide
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-3-(4-methylpiperazin-1-yl)propanamide
1-{2-[4-(2-phenylpropyl)-1H-1,2,3-triazol-1-yl]ethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
N-[4-(1-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-1H-imidazol-2-yl)phenyl]acetamide
4-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-7-methyl-3,4-dihydro-2H-1,4-benzothiazin-3-one
3-{1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]pyrrolidin-2-yl}-5-methyl-1,2-oxazole
3-{2-[(4-fluoro-2-methylphenyl)carbamoyl]ethyl}-N-(2-methoxyethyl)piperidine-1-carboxamide
2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}acetamide
3-(2-amino-1,3-thiazol-4-yl)-1-[4-(benzyloxy)piperidin-1-yl]propan-1-one
2-methyl-5-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
[1-({1-[(1-methyl-5-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanamine
methyl 4-({[1-(pyridin-3-ylmethyl)piperidin-4-yl]carbamoyl}amino)benzoate
1-(1-cyclobutanecarbonylpiperidin-4-yl)-2-(3,4-dimethoxyphenyl)-5-fluoro-1H-1,3-benzodiazole
7-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}-3-methyl-3,4-dihydroquinazolin-4-one
N-[3-(3-fluorophenyl)phenyl]-1-[(3-hydroxy-4-methoxyphenyl)methyl]piperidine-4-carboxamide
3-{2-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
7-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-2,7-diazaspiro[4.4]nonane-1,3-dione
2-amino-4-[2-(4-methoxyphenyl)pyrimidin-5-yl]-7-methyl-5H,7H-furo[3,4-b]pyridine-3-carbonitrile
N-({[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]carbamoyl}methyl)propanamide
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
[4-({1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]pyrrolidin-3-yl}methyl)phenyl]methanol
3-[(4aR,7aS)-4-[(4-chlorophenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
N-[2-(4-chlorophenyl)propyl]-2,4-dimethyl-1,3-oxazole-5-carboxamide
3-(2,3-dihydro-1H-inden-4-yl)-1-[(5-methylpyrazin-2-yl)methyl]urea
2-[1-(4,6-dimethylpyrimidin-2-yl)-1H-pyrazol-4-yl]-7-methoxy-N,N-dimethylquinoline-4-carboxamide
N-cyclopropyl-3-[5-(1-ethylpyrrolidine-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide