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1-(3-cyano-4-ethoxyphenyl)-3-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}urea
N,N,4-trimethyl-3-({methyl[(methylcarbamoyl)methyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-(4-{[(2S)-1-methylpyrrolidin-2-yl]methyl}-1,4-diazepan-1-yl)-1,3-benzothiazole
1-(2-methylpropyl)-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide
[(3-{[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(naphthalen-1-ylmethyl)amine
3-(1-butyl-1H-pyrazol-5-yl)-1-{1-oxaspiro[4.4]nonan-3-yl}urea
2-{5-[2-chloro-5-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-{[4-(aminomethyl)phenyl]methyl}-2-(dimethylamino)-2-(3-methylphenyl)acetamide
2,5-dimethyl-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-[(3S)-2-oxoazepan-3-yl]-4-(quinolin-6-yloxy)piperidine-4-carboxamide
1-[2-({2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)ethyl]imidazolidin-2-one
2-{1-[(2-ethoxyphenyl)methyl]-4-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
methyl 3-(cyclobutylmethoxy)-5-(4-ethylpiperazine-1-carbonyl)benzoate
methyl 1-(cyclopropylmethyl)-2-oxo-3-[3-(1H-pyrazol-1-yl)propyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
2-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-(propan-2-yl)acetamide
N-[(2-methoxyphenyl)methyl]-2-{[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]amino}acetamide
1-[1-(3-fluorobenzoyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
N-[(3-chlorophenyl)methyl]-3-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}propanamide
methyl 3-[(cyclohexylformamido)methyl]-5-(2-methoxybenzamido)benzoate
1,5,6-trimethyl-2-oxo-N-[(3,4,5-trimethoxyphenyl)methyl]-1,2-dihydropyridine-3-carboxamide
5-{2-[2-(2,4-dimethoxyphenyl)-1H-imidazol-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{[(2R)-1-ethylpyrrolidin-2-yl]methyl}-4-(2-phenylethyl)-1H-1,2,3-triazole
N-benzyl-4-(5-{[(2-methoxyphenyl)carbamoyl]amino}-1H-pyrazol-1-yl)piperidine-1-carboxamide
2-{[2-(morpholine-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}quinolin-4-ol
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-(butan-2-yl)-N3-ethyl-N5-(furan-2-ylmethyl)-N3-(2-methylprop-2-en-1-yl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-({2-[1-(pyrrolidine-1-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-(furan-2-ylmethyl)-2,7-dioxo-N-(pyridin-4-ylmethyl)-1,3-diazepane-4-carboxamide
1-[(2-chloro-4-hydroxyphenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
methyl[(3-methylphenyl)methyl]{[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}amine
4-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-2-(trifluoromethyl)morpholine
4-(3,4-dimethoxybenzoyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
2-{4-[(2-methyl-1,3-thiazol-5-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
2-[1-(1-methylpiperidin-4-yl)-4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperazin-2-yl]ethan-1-ol
2-(1-benzyl-4-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl)ethan-1-ol
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
3-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-4H-pyrido[1,2-a]pyrimidin-4-one
N-({2-[4-(piperidine-1-sulfonyl)phenyl]phenyl}methyl)propanamide
methyl 5-[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
2-(oxan-2-ylmethyl)-2,3-dihydro-1,2-benzothiazol-3-one
N-[(3R,7S,8aS)-3-[(benzylsulfanyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-chlorobenzamide
7-(5-chloropyridin-2-yl)-4-(oxolan-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[2-methoxy-5-(1,2-oxazinan-2-ylmethyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
N-methyl-3-(2-oxoimidazolidin-1-yl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]benzamide
1-[7-(1,2,3,4-tetrahydroquinoline-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]propan-1-one
N,N-dimethyl-2-[(1S,5R)-3-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
({3-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)diethylamine
2-[1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)pyrrolidin-2-yl]-6-methyl-1H-1,3-benzodiazole
2-(2-fluorophenoxymethyl)-N-[2-(6-methylpyridin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
5-(oxolan-2-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]thiophene-2-carboxamide