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1-[2-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propan-1-one
1-(3-propyl-1H-pyrazole-5-carbonyl)-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
2-{3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-5-methoxy-1,4-dihydropyridin-4-one
8-[(4-fluoro-2-methylphenyl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
3-[1-(cyclohex-1-ene-1-carbonyl)piperidin-3-yl]-N-[(2,4-dimethoxyphenyl)methyl]propanamide
N-{5H,6H,7H,8H,9H,10H,11H-cycloocta[b]indol-2-ylmethyl}-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
N-(4-{2-[(1R,4R)-2-azabicyclo[2.2.1]heptan-2-yl]acetamido}phenyl)-5-methylfuran-3-carboxamide
1-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
1-{1'-[(4-methoxy-3-methylphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
2-[4-(2-phenylazetidine-1-carbonyl)piperidin-1-yl]acetamide
ethyl 1-(3-methylfuran-2-carbonyl)-4-(2-phenylethyl)piperidine-4-carboxylate
N-(2-methoxyethyl)-3-({1-[4-(1H-pyrazol-1-yl)butan-2-yl]piperidin-4-yl}oxy)benzamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methylacetamide
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-N-methyl-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
4-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1-(prop-2-en-1-yl)pyrrolidin-2-one
2-{1-methyl-4-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
1-{1-[(3-fluorophenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
3-{[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]sulfamoyl}-N-(2-methylpropyl)benzamide
2-(adamantan-1-yl)-N-(3-ethoxypropyl)acetamide
ethyl 4-(cyclopropylmethyl)-1-[2-(morpholin-4-yl)-2-(pyridin-3-yl)acetyl]piperidine-4-carboxylate
1-(3,4-dimethylphenyl)-N-(6-methylpyridazin-3-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-3-methoxypiperidine
N,5-dimethyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-1,3-oxazole-4-carboxamide
6-(methoxymethyl)-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]pyrimidin-4-amine
(3S)-N-tert-butyl-2-(pyrrolidine-1-carbonyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
4-(4-{[3-(2-hydroxyethyl)-4-(thiophen-2-ylmethyl)piperazin-1-yl]methyl}phenyl)but-3-yn-1-ol
8-methoxy-2-methyl-5-{2-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}quinoline
5-amino-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-1H-pyrazole-3-carboxamide
2-(2-hydroxyethyl)-8-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one
N-methyl-5-{3-[(propan-2-yl)carbamoyl]benzenesulfonamidomethyl}-1,2,4-oxadiazole-3-carboxamide
2-methoxy-6-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
2-methoxy-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]acetamide
3-(3-{1-[(4-methyl-1,3-thiazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridine
N-[(3S)-piperidin-3-yl]-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2,2-diphenyl-1-[4-(pyridin-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]ethan-1-ol
3-{2-[({4-[3-(4-ethylpiperazin-1-yl)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)amino]ethyl}-1,3-oxazolidin-2-one
7-(4,4,4-trifluorobutanoyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-amino-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)-4-[5-(1H-pyrazol-3-yl)furan-2-yl]pyridine-3-carbonitrile
1-(3-oxo-3-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}propyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(methanesulfonylmethyl)-1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]piperidine
2-(4-fluorophenyl)-1-[(4-methanesulfonylphenyl)methyl]piperidine
N-({1-[(2-aminopyrimidin-5-yl)methyl]piperidin-3-yl}methyl)-4-phenylbenzamide
N-({2-[(dimethylamino)methyl]phenyl}methyl)-6-methoxypyrimidin-4-amine
(3R,4R)-4-[({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)amino]pyrrolidin-3-ol
(2R)-2-amino-3-(1H-indol-3-yl)-1-[3-(3-methylphenoxy)azetidin-1-yl]propan-1-one
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[1-(methoxymethyl)cyclopropanecarbonyl]piperidine
2-(1-methylcyclopropanecarbonyl)-N-(2-phenoxyethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
1-{3-[3-(2-methoxyethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]phenyl}-5-methyl-1H-1,2,3,4-tetrazole
1-[1-(furan-2-yl)ethyl]-4-[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]-1H-1,2,3-triazole
4-[(6-amino-2-methylpyrimidin-4-yl)amino]-1-(3-methoxyphenyl)pyrrolidin-2-one