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2-{3,5-dimethyl-4-[(1E)-pent-1-en-1-yl]-1H-pyrazol-1-yl}acetic acid
3-methyl-7-[(5-methylnaphthalen-1-yl)methyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
4-[(4-methoxynaphthalen-1-yl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(benzyloxy)-N-[2-(2-methoxyethoxy)phenyl]piperidine-1-carboxamide
5-{5-[4-(1H-imidazol-1-yl)phenyl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
2-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]benzamide
7-(3-chlorophenyl)-4-[(2-hydroxy-3-methylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N,N-dimethyl-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]aniline
N-[(3S,4R)-4-hydroxyoxolan-3-yl]-N-methyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
5-chloro-3-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}-1,2-dihydropyridin-2-one
N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
8-[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazole-4-carbonyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
(2S)-3-(4-hydroxyphenyl)-2-[(1-methyl-4-oxo-1,4-dihydroquinolin-3-yl)formamido]propanamide
N-(1-cycloheptylpiperidin-3-yl)-3-(3,5-dimethyl-1H-pyrazol-1-yl)propanamide
8-[6-methyl-2-(methylamino)pyrimidin-4-yl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
ethyl 3-[(3-methoxyphenyl)methyl]-1-(pyridin-4-ylmethyl)piperidine-3-carboxylate
3-[2-(dimethylsulfamoyl)ethyl]-1-(2-methoxypyridin-3-yl)urea
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[1-(pyridin-3-yl)propan-2-yl]amine
{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)methylamine
N-cyclopropyl-1-{2-[1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)piperidin-2-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
1-(2-hydroxyethyl)-N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}piperidine-4-carboxamide
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)propanamide
5-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}-2,3-dihydro-1H-pyrazol-3-one
N,N-dimethyl-3-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamido]azepane-1-carboxamide
5-chloro-N-[2-(dimethylamino)ethyl]-N,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-[(2R,3R,6R)-5-[2-(methylamino)-1,3-thiazole-4-carbonyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-(2,4-dimethoxyphenyl)-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,2,4-triazin-3-amine
3-ethyl-4-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-5-methyl-1,2-oxazole
({6-[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]-2-methylpyrimidin-4-yl}methyl)dimethylamine
N-methyl-4-({methyl[(3-methylpyridin-2-yl)methyl]amino}methyl)benzene-1-sulfonamide
2-amino-4-(5-cyano-1-ethyl-1H-pyrrol-3-yl)-6-(3,5-dimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
2-[3-cyclopentyl-5-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
3-[2-(2-fluorophenoxy)pyridin-3-yl]-1-[2-(4-hydroxypiperidin-1-yl)ethyl]urea
5-(furan-3-ylmethyl)-11-methyl-8-thia-3,5,10-triazatricyclo[7.4.0.02,7]trideca-1(13),2(7),3,9,11-pentaen-6-one
1-[1-(2-fluorobenzoyl)piperidin-4-yl]-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-ethyl-1-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[1-(methoxymethyl)cyclobutanecarbonyl]-4-(2-methoxyphenoxy)piperidine
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
4-[(3-chloro-4-hydroxy-5-methoxyphenyl)methyl]-1-[(3-methylphenyl)methyl]piperazin-2-one
{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}[1-(1H-imidazol-1-yl)propan-2-yl]amine
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-cyclopropylacetamide
N2,N2,N4,N4-tetramethyl-7-[2-(methylamino)pyridine-3-carbonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
2-(methylamino)-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]acetamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-1,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-{2-[2-(6-chloro-2-fluoro-3-methylphenyl)-1H-imidazol-1-yl]ethyl}imidazolidin-2-one
1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(morpholin-3-yl)ethan-1-one
(1R,5S,6R)-3-cyclopentyl-N-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
2-amino-1-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one