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1-(1,4-diazepan-1-yl)-2-(2-propyl-1H-1,3-benzodiazol-1-yl)propan-1-one
2-(adamantan-1-yl)-4-hydroxy-N-[2-(pyridin-3-yl)ethyl]pyrimidine-5-carboxamide
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-ethyl-1H-1,2,4-triazole
2-chloro-4-({4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-6-methoxyphenol
N-[3-(2-methoxyphenyl)propyl]thiolan-3-amine
3-({[(2-aminopyrimidin-5-yl)methyl](methyl)amino}methyl)-N-(2-methyl-2H-1,2,3-triazol-4-yl)benzamide
3-(3-fluorophenyl)-N-(piperidin-4-yl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
5-methyl-N-[2-(pyridin-2-yl)ethyl]-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
2-[(4aR,7aS)-6,6-dioxo-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
(3S,4R)-4-methyl-1-[1-(4-methylbenzoyl)piperidine-4-carbonyl]piperidine-3,4-diol
2-butyl-8-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]-2,8-diazaspiro[5.5]undecan-3-one
2-{4-[2-(3-fluorophenyl)azepane-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
N-[2-(oxan-2-yl)ethyl]-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
(3S,5R)-1-(5-methylhexanoyl)-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
4-(4-{[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]amino}piperidin-1-yl)-N,N-dimethylbenzamide
4-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl](methyl)sulfamoyl}-N-methylthiophene-2-carboxamide
2-[1-({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)piperidin-2-yl]pyridine
2-[1-methyl-5-(3-methyl-1-phenyl-1H-pyrazol-4-yl)-1H,4H-pyrazolo[3,4-d]imidazol-3-yl]pyridine
6-oxo-N-(pyrimidin-4-ylmethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
N-{1-[1-(2-hydroxyethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
8-chloro-2-(furan-2-yl)-4-(1,4-oxazepane-4-carbonyl)quinoline
[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)methylamine
4-(3-{4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}butyl)phenol
3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)propanamide
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
1-methyl-4-[5-(2-methyloxolane-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl]piperazine
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-1-(pyrimidin-2-yl)piperidin-4-amine
5-methyl-2-[2-(morpholin-4-ylmethyl)-1,4-oxazepane-4-carbonyl]phenol
1-{[6-(3-fluoro-4-methoxyphenyl)pyridin-3-yl]methyl}-4-methylpiperazine
3-({2-[2-(9H-fluoren-2-yl)-1H-imidazol-1-yl]ethyl}sulfanyl)-4-methyl-4H-1,2,4-triazole
N-[(3R,4S)-1-(5,6-dimethylpyrazin-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]-4-methylpiperidine-4-carboxamide
N-{1-[1-(3-methoxy-2,2-dimethylpropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide
1-{1'-[3-(dimethylamino)pyrazin-2-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
methyl 5-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}-5-oxopentanoate
2-methyl-4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-6-(1H-pyrazol-1-yl)pyrimidine
4-[4-(3,5-difluoropyridine-2-carbonyl)-5-methyl-2-oxopiperazin-1-yl]benzonitrile
1-{2-[({[3-(methylsulfanyl)phenyl]methyl}amino)methyl]phenoxy}-3-(thiomorpholin-4-yl)propan-2-ol
ethyl 5-methyl-1-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
3-[(3R,4S)-1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
3-{[(2-methylpropyl)(thiophen-3-ylmethyl)amino]methyl}pyrrolidin-3-ol
4-(1H-imidazol-1-yl)-N-[(4-methanesulfonylmorpholin-2-yl)methyl]benzamide
1-(dimethylsulfamoyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(3S,4R)-3-methoxy-1-(3-phenoxybenzoyl)piperidin-4-amine
1-({2-methoxy-5-[(2-phenylazetidin-1-yl)methyl]phenyl}methyl)-1H-1,2,4-triazole
2-[(2-fluorophenyl)methyl]-4-{4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
[1-(2-amino-5-butyl-6-methylpyrimidin-4-yl)piperidin-3-yl]methanol
3-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-ethylphenyl)urea